SCHEMBL6301116

SCHEMBL6301116

CCCCNC(=O)c1ccc(N2CCC(NCCC(O)Oc3cccc(N)c3N)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASR P41180 8/20 0.41
HDAC3 O15379 4/20 0.40
HDAC1 Q13547 3/20 0.40
KDM4E B2RXH2 2/20 0.40
CHRM2 P08172 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM3 P20309 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADRB3 P13945 2/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
POLB P06746 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
CHRNA10 Q9GZZ6 1/20 0.38
CHRNA9 Q9UGM1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6303593 0.89 CASR (0.39) CASRKDM4ECHRM2CHRM5CHRM3
SCHEMBL6309219 0.86 ADRB1 (0.39) KDM4ECHRM2CHRM5CHRM3ALDH1A1
SCHEMBL6301113 0.85 ADRB3 (0.43) CASRHDAC3HDAC1ADRB3ADRB2
SCHEMBL6301068 0.83 ADRB3 (0.45) CASRKDM4ECHRM2CHRM5CHRM3
SCHEMBL6308617 0.75 MAPT (0.40) ALDH1A1SMN1; SMN2ADRB3ADRB2ADRB1
SCHEMBL6303591 0.74 ADRB3 (0.42) CASRALDH1A1SMN1; SMN2ADRB3ADRB2
SCHEMBL6301416 0.72 SMYD3 (0.54) HDAC3HDAC1ALDH1A1SMN1; SMN2POLB
Water SCHEMBL5211069 0.71 SMYD3 (0.53) HDAC3HDAC1ALDH1A1SMN1; SMN2POLB
SCHEMBL6301065 0.70 ADRB3 (0.61) CASRADRB3ADRB2ADRB1
Hydrochloric Acid SCHEMBL6139757 0.70 SMYD3 (0.52) HDAC3HDAC1ALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6858629-B1 Heteroaryloxy propanolamines, preparation method and pharmaceutical compositions containing same SANOFI-SYNTHELABO (FR) 2005-02-22 US disclosed
EP-1214313-B1 HETEROARYLOXY PROPANOLAMINES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI SYNTHELABO (FR) 2004-06-30 EP disclosed