SCHEMBL630338

SCHEMBL630338

CCOC(=O)C1=CCCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.49
ATM Q13315 1/20 0.44
GPR119 Q8TDV5 3/20 0.42
GLA P06280 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
USP2 O75604 1/20 0.41
ESR2 Q92731 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
NR1H2 P55055 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6218755 0.89 ADORA1 (0.49) ADORA1ATMGPR119GLASMN1; SMN2
SCHEMBL12931062 0.88 ADORA1 (0.53) ADORA1GPR119GLASMN1; SMN2NPSR1
SCHEMBL26134595 0.86 CHRM3 (0.48) GPR119SMN1; SMN2MEN1ALDH1A1LMNA
SCHEMBL6541860 0.82 ADORA1 (0.47) ADORA1ATMGPR119GLASMN1; SMN2
SCHEMBL31195159 0.80 ADORA1 (0.48) ADORA1ATMGPR119GLASMN1; SMN2
SCHEMBL15894090 0.80 USP2 (0.47) GPR119SMN1; SMN2MEN1ALDH1A1LMNA
SCHEMBL13496714 0.79 USP2 (0.46) ATMGPR119SMN1; SMN2MEN1ALDH1A1
SCHEMBL6958805 0.78 ADORA1 (0.48) ADORA1ATMGPR119GLASMN1; SMN2
SCHEMBL2081926 0.78 ADORA1 (0.51) ADORA1ATMGPR119SMN1; SMN2NPSR1
SCHEMBL12923869 0.78 ADORA1 (0.51) ADORA1ATMGPR119SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250223277-A1 COMPLEMENT FACTOR B INHIBITORS AND USES THEREOF NOVARTIS PHARMA AG (CH) 2025-07-10 US disclosed
CN-119137099-A Complement factor B inhibitors and uses thereof 诺华股份有限公司 2024-12-13 CN disclosed
WO-2023187715-A1 COMPLEMENT FACTOR B INHIBITORS AND USES THEREOF NOVARTIS AG (CH) 2023-10-05 WO disclosed
US-11584765-B2 Polycyclic amines as sigma receptor modulators Ecstasy LLC (US) 2023-02-21 US disclosed
CN-110662541-B Polycyclic amines as opioid receptor modulators 王晓冬 2023-02-10 CN disclosed
US-20220411442-A1 POLYCYCLIC AMINES AS OPIOID RECEPTOR MODULATORS Ecstasy LLC 2022-12-29 US disclosed
EP-3398598-B1 SULFONAMIDE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF HITGEN INC (CN) 2022-04-06 EP disclosed
US-11149008-B2 Sulfamide derivatives and preparation method and use thereof HitGen, Inc. 2021-10-19 US disclosed
CN-106928198-B Sulfonamide derivative and preparation method and application thereof 成都先导药物开发股份有限公司 2020-07-28 CN disclosed
US-10676456-B2 Polycyclic amines as opioid receptor modulators Ecstasy LLC 2020-06-09 US disclosed
EP-2420234-B1 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION AS PARP INHIBITORS FOR USE IN TREATING CANCER ABBOTT LAB (US) 2013-07-10 EP disclosed
EP-2420499-B1 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION AS POTENT PARP INHIBITORS ABBOTT LAB (US) 2013-07-10 EP disclosed
WO-2013025425-A1 SOLUBLE GUANYLATE CYCLASE ACTIVATORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-21 WO disclosed
EP-1869011-B1 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LAB (US) 2012-08-01 EP disclosed
EP-2420234-A1 1H-benzimidazole-4-carboxamides substituted with a quaternary carbon at the 2-position as PARP inhibitors for use in treating cancer Abbott Laboratories (US) 2012-02-22 EP disclosed
EP-2420499-A1 1H-benzimidazole-4-carboxamides substituted with a quaternary carbon at the 2-position as potent PARP inhibitors Abbott Laboratories (US) 2012-02-22 EP disclosed
US-7550603-B2 1H-benzimidazole-4-carboxamides substituted with a quaternary carbon at the 2-position are potent PARP inhibitors ABBOTT LABORATORIES INC. (US) 2009-06-23 US disclosed
EP-1869011-A2 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LABORATORIES (US) 2007-12-26 EP disclosed
WO-2006110816-A2 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH A QUATERNARY CARBON AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LABORATORIES (US) 2006-10-19 WO disclosed
US-20060229289-A1 1H-benzimidazole-4-carboxamides substituted with a quaternary carbon at the 2-position are potent PARP inhibitors ABBVIE INC. 2006-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10676456-B2 Polycyclic amines as opioid receptor modulators OPRM1, OPRL1, OPRK1 ADORA1 144/4885ATM 4130/4885GPR119 354/4885
US-11584765-B2 Polycyclic amines as sigma receptor modulators OPRM1, SIGMAR1, OPRK1 ADORA1 77/4885ATM 4020/4885GPR119 385/4885
US-20250223277-A1 COMPLEMENT FACTOR B INHIBITORS AND USES THEREOF CFB, CFH, C1QBP ADORA1 3280/4885ATM 3156/4885GPR119 2495/4885
US-11149008-B2 Sulfamide derivatives and preparation method and use thereof HDAC6, HDAC1, HDAC11 ADORA1 4138/4885ATM 3952/4885GPR119 762/4885
US-20060229289-A1 1H-benzimidazole-4-carboxamides substituted with a quaternary carbon at the 2-position are potent PARP inhibitors PARP1, PARP2, PARP4 ADORA1 3607/4885ATM 531/4885GPR119 3493/4885
US-20220411442-A1 POLYCYCLIC AMINES AS OPIOID RECEPTOR MODULATORS OPRM1, OPRL1, OPRK1 ADORA1 144/4885ATM 4130/4885GPR119 354/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.