SCHEMBL6306196

SCHEMBL6306196

Cc1ccccc1-c1nc2ccccc2c(=O)n1CCCN

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASR P41180 2/20 0.53
TSHR P16473 2/20 0.52
TDP1 Q9NUW8 5/20 0.51
RXRA P19793 2/20 0.51
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TP53 P04637 1/20 0.51
MAPT P10636 3/20 0.50
PTK2B Q14289 1/20 0.48
GAA P10253 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313293 0.88 CASR (0.52) CASRTDP1RXRA
SCHEMBL6308910 0.87 CASR (0.53) CASRTSHRTDP1RXRAALDH1A1
SCHEMBL6313246 0.86 CASR (0.58) CASRSMN1; SMN2TP53MAPTMEN1
SCHEMBL6308902 0.86 EGFR (0.64) CASRSMN1; SMN2TP53MAPTMEN1
SCHEMBL6307828 0.84 F11 (0.52) TSHRTDP1RXRAALDH1A1SMN1; SMN2
SCHEMBL6309029 0.84 CASR (0.68) CASRTSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL5921199 0.83 CASR (0.75) CASRSMN1; SMN2GAAMEN1KMT2A
SCHEMBL6314431 0.82 MEN1 (0.67) CASRALDH1A1TP53MAPTGAA
SCHEMBL6314002 0.82 CASR (0.65) CASRTSHRALDH1A1SMN1; SMN2TP53
SCHEMBL6306167 0.80 KMT2A (0.63) CASRTSHRALDH1A1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed