SCHEMBL6307635

SCHEMBL6307635

NCCCn1c(CCc2ccccc2)nc2cc(Cl)ccc2c1=O

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.57
KIF11 P52732 4/20 0.52
CYP3A4 P08684 2/20 0.52
GHSR Q92847 5/20 0.47
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
MAP1LC3B Q9GZQ8 1/20 0.45
CYP2C19 P33261 1/20 0.45
KCNH2 Q12809 1/20 0.45
CASR P41180 2/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6309838 0.92 CASR (0.53) EGFRKIF11CYP3A4GHSRPDE4A
SCHEMBL6309040 0.87 PDE4A (0.56) GHSRPDE4APDE4BPDE4CPDE4D
SCHEMBL6313871 0.83 KIF11 (0.51) EGFRKIF11CYP3A4PDE4APDE4B
SCHEMBL6313933 0.81 GHSR (0.52) GHSRPDE4APDE4BPDE4CPDE4D
SCHEMBL6314890 0.81 EGFR (0.86) EGFRCASR
SCHEMBL6314802 0.79 EGFR (0.83) EGFRCASR
SCHEMBL6313515 0.78 GHSR (0.50) GHSRMEN1KMT2A
SCHEMBL5878284 0.78 EGFR (0.45) EGFRKIF11CYP3A4PDE4APDE4B
SCHEMBL7546931 0.77 MEN1 (0.60) EGFRMEN1KMT2A
SCHEMBL7546935 0.77 MEN1 (0.60) EGFRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed