SCHEMBL6313933

SCHEMBL6313933

Cc1ccc2nc(CCc3ccccc3)n(CCCN)c(=O)c2c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 5/20 0.52
CASR P41180 1/20 0.46
DHFR P00374 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
PLK1 P53350 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6309838 0.86 CASR (0.53) GHSRCASRPDE4APDE4BPDE4C
SCHEMBL6313515 0.86 GHSR (0.50) GHSRMEN1KMT2A
SCHEMBL6309040 0.86 PDE4A (0.56) GHSRCASRMEN1KMT2APDE4A
SCHEMBL6308411 0.82 DHFR (0.49) DHFRPDE4APDE4BPDE4CPDE4D
SCHEMBL6307779 0.81 EGFR (0.57) CASRMEN1KMT2A
SCHEMBL6307635 0.81 EGFR (0.57) GHSRCASRMEN1KMT2APDE4A
SCHEMBL6394256 0.79 EGFR (0.55) GHSRCASRMEN1KMT2A
SCHEMBL6313293 0.78 CASR (0.52) GHSRCASRDHFR
SCHEMBL6308112 0.78 KMT2A (0.50) GHSRCASRKMT2A
SCHEMBL5877934 0.77 GHSR (0.41) GHSRDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed