SCHEMBL6308352

SCHEMBL6308352

NCc1cccc(Cn2c(CCc3ccccc3)nc3ccccc3c2=O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.59
PDE4B Q07343 2/20 0.59
PDE4C Q08493 2/20 0.59
PDE4D Q08499 2/20 0.59
TLR8 Q9NR97 1/20 0.53
TLR7 Q9NYK1 1/20 0.53
RAB9A P51151 2/20 0.50
POLB P06746 1/20 0.50
ALDH1A1 P00352 5/20 0.49
LMNA P02545 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
RECQL P46063 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CASR P41180 2/20 0.47
F11 P03951 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
CYP1A2 P05177 1/20 0.44
GAA P10253 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313871 0.89 KIF11 (0.51) PDE4APDE4BPDE4CPDE4DTLR8
SCHEMBL6308411 0.88 DHFR (0.49) PDE4APDE4BPDE4CPDE4D
SCHEMBL6309834 0.88 PTGES (0.50) PDE4APDE4BPDE4CPDE4DRAB9A
SCHEMBL28206539 0.87 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DRAB9A
SCHEMBL6313964 0.85 CYP1A2 (0.52) PDE4APDE4BPDE4CPDE4DTLR8
SCHEMBL6309810 0.81 ALDH1A1 (0.76) RAB9APOLBALDH1A1LMNASMN1; SMN2
SCHEMBL6306194 0.80 ALDH1A1 (0.72) RAB9APOLBALDH1A1LMNASMN1; SMN2
SCHEMBL6306807 0.79 ALDH1A1 (0.56) PDE4APDE4BPDE4CPDE4DTLR8
SCHEMBL6309040 0.79 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DRAB9A
SCHEMBL6308509 0.78 ALDH1A1 (0.65) RAB9AALDH1A1LMNASMN1; SMN2RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed