SCHEMBL6314477

SCHEMBL6314477

CSc1nc(N)nc(-c2cccnc2)n1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.69
HSP90AB1 P08238 2/20 0.69
SMN1; SMN2 Q16637 2/20 0.60
TSHR P16473 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
ADORA2A P29274 5/20 0.51
ADORA1 P30542 5/20 0.51
LMNA P02545 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HTT P42858 2/20 0.46
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP2A6 P11509 3/20 0.44
PTK2 Q05397 1/20 0.44
POLB P06746 2/20 0.43
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23092286 0.83 SMN1; SMN2 (0.70) HSP90AA1HSP90AB1SMN1; SMN2TSHRNPSR1
SCHEMBL30740045 0.83 SMN1; SMN2 (0.70) HSP90AA1HSP90AB1SMN1; SMN2TSHRNPSR1
SCHEMBL9489052 0.83 SMN1; SMN2 (0.70) HSP90AA1HSP90AB1SMN1; SMN2TSHRNPSR1
SCHEMBL4093530 0.82 HSP90AA1 (1.00) HSP90AA1HSP90AB1TSHRNPSR1ADORA2A
SCHEMBL11192075 0.81 ALDH1A1 (0.46) HSP90AA1HSP90AB1SMN1; SMN2TSHRNPSR1
SCHEMBL14523587 0.79 SMN1; SMN2 (0.65) HSP90AA1HSP90AB1SMN1; SMN2TSHRNPSR1
SCHEMBL15614062 0.78 ADORA2A (0.64) HSP90AA1HSP90AB1SMN1; SMN2TSHRNPSR1
SCHEMBL6313572 0.74 HSP90AA1 (0.67) HSP90AA1HSP90AB1ADORA2AADORA1HTT
SCHEMBL6309967 0.73 HSP90AA1 (0.72) HSP90AA1HSP90AB1SMN1; SMN2NPSR1ADORA2A
SCHEMBL5032444 0.73 SMN1; SMN2 (0.73) SMN1; SMN2TSHRNPSR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6919339-B2 ABCA-1 elevating compounds CV THEAPEUTICS, INC. (US) 2005-07-19 US disclosed
US-20020128266-A1 ABCA-1 elevating compounds CV THERAPEUTICS, INC. 2002-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020128266-A1 ABCA-1 elevating compounds ABCD3, ABCE1, ABCB4 HSP90AA1 1676/4885HSP90AB1 1191/4885SMN1; SMN2 4558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.