SCHEMBL6314846

SCHEMBL6314846

CCOC(=O)c1cnc(N(C)c2cc3c(cc2C)C(C)C(C)CC3(C)C)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 7/20 0.41
RXRB P28702 6/20 0.41
RXRG P48443 6/20 0.41
PPARG P37231 1/20 0.41
NR1H3 Q13133 1/20 0.41
RARA P10276 3/20 0.35
RARB P10826 3/20 0.35
RARG P13631 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP3A4 P08684 1/20 0.35
P2RY12 Q9H244 2/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5180347 0.82 RXRA (0.59) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5178703 0.69 RXRA (0.65) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5179745 0.69 RXRA (0.61) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5179721 0.69 RXRA (0.58) RXRARXRBRXRGPPARGNR1H3
SCHEMBL10844326 0.69 RARB (0.48) RXRARXRBRXRGRARARARB
SCHEMBL10844308 0.69 RARB (0.48) RXRARXRBRXRGRARARARB
SCHEMBL5179533 0.67 RXRA (0.72) RXRARXRBRXRGPPARGNR1H3
SCHEMBL11530672 0.66 ALDH1A1 (0.56) CYP3A4CYP2C9CYP2C19ALDH1A1NPSR1
SCHEMBL501775 0.65 RXRA (0.52) RXRARXRBRXRGPPARGNR1H3
SCHEMBL5178994 0.64 CYP2C9 (0.40) KMT2AP2RY12CYP2C9CYP2C19HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6869959-B1 Heterocyclic carboxylic acid derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN INC. (JP) 2005-03-22 US disclosed