SCHEMBL6314997

SCHEMBL6314997

COc1ccc(-c2nc(CC(=O)NO)oc2-c2ccc(S(N)(=O)=O)cc2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.52
PTGS1 P23219 15/20 0.52
CDK2 P24941 1/20 0.47
MEP1B Q16820 1/20 0.47
ABCB11 O95342 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6315576 0.89 PTGS2 (0.50) PTGS2PTGS1ALDH1A1
SCHEMBL8549849 0.87 PTGS2 (0.57) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6315415 0.87 PTGS2 (0.50) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL5732493 0.87 PTGS2 (0.51) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6315005 0.85 PTGS2 (0.45) PTGS2PTGS1CDK2MEP1B
SCHEMBL6314953 0.84 CA9 (0.49) PTGS2PTGS1CDK2MEP1BALDH1A1
SCHEMBL7505035 0.84 PTGS2 (0.57) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6309705 0.83 PTGS1 (0.46) PTGS2PTGS1
SCHEMBL6315584 0.83 PTGS2 (0.51) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6308685 0.83 PTGS2 (0.60) PTGS2PTGS1MEP1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6875785-B2 Heterocyclo substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors PHARMACIA CORPORATION (US) 2005-04-05 US claimed