SCHEMBL6326353

SCHEMBL6326353

O=C(NCCCNc1n[nH]c(=O)c2cccnc12)NC1CC1c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
BMP1 P13497 2/20 0.39
DYRK1A Q13627 2/20 0.39
CLK2 P49760 1/20 0.39
CLK3 P49761 1/20 0.39
WNT1 P04628 1/20 0.39
SIRT5 Q9NXA8 1/20 0.38
MAPK1 P28482 3/20 0.38
P2RX7 Q99572 3/20 0.38
AURKB Q96GD4 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PAK4 O96013 1/20 0.36
CNR1 P21554 1/20 0.36
KDM1A O60341 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6327259 0.77 MTNR1A (0.44) MAPK1AURKB
SCHEMBL6473156 0.76 PARP1 (0.45) AURKBSMN1; SMN2
SCHEMBL6323949 0.76 ALDH1A1 (0.44) MAPK1AURKB
SCHEMBL5076368 0.71 PARP1 (0.45)
SCHEMBL5074298 0.71 MEN1 (0.35) MAPK1AURKB
SCHEMBL5076362 0.70 PARP1 (0.45) MAPK1AURKB
SCHEMBL5077387 0.69 KAT2B (0.35) MAPK1
SCHEMBL6328281 0.68 GAA (0.49) MAPK1SMN1; SMN2
SCHEMBL6334650 0.68 ALDH1A1 (0.44) MAPK1AURKB
SCHEMBL5074305 0.66 MEN1 (0.35) MAPK1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924284-B2 PARP inhibitors ICOS CORPORATION (US) 2005-08-02 US disclosed