SCHEMBL6327259

SCHEMBL6327259

CC(=O)NCCCNc1n[nH]c(=O)c2cccnc12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.44
PARP1 P09874 7/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
KAT2B Q92831 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
TSHR P16473 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
AURKB Q96GD4 1/20 0.37
MTNR1B P49286 1/20 0.37
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6323949 0.89 ALDH1A1 (0.44) PARP1ALDH1A1MAPK1KAT2BHDAC1
SCHEMBL6473156 0.82 PARP1 (0.45) PARP1L3MBTL1ALDH1A1KAT2BTSHR
SCHEMBL5076368 0.82 PARP1 (0.45) PARP1KAT2B
SCHEMBL5077387 0.81 KAT2B (0.35) PARP1ALDH1A1MAPK1KAT2BHDAC1
SCHEMBL5076362 0.80 PARP1 (0.45) PARP1ALDH1A1MAPK1KAT2BAURKB
SCHEMBL6334650 0.80 ALDH1A1 (0.44) MTNR1AL3MBTL1ALDH1A1MAPK1KAT2B
SCHEMBL6326353 0.77 EPHX2 (0.41) MAPK1AURKB
SCHEMBL6328281 0.76 GAA (0.49) ALDH1A1MAPK1
SCHEMBL5074298 0.75 MEN1 (0.35) PARP1MAPK1CYP1A2AURKB
SCHEMBL6333338 0.72 LMNA (0.48) ALDH1A1MAPK1HDAC1TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924284-B2 PARP inhibitors ICOS CORPORATION (US) 2005-08-02 US disclosed