SCHEMBL6327688

SCHEMBL6327688

O=C1Cc2ccccc2N1c1ccc(Cl)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.74
KMT2A Q03164 5/20 0.51
MEN1 O00255 4/20 0.51
DRD2 P14416 2/20 0.51
DRD5 P21918 1/20 0.51
DRD3 P35462 1/20 0.51
TNKS O95271 1/20 0.49
OPRK1 P41145 1/20 0.49
PDE4D Q08499 1/20 0.49
DRD4 P21917 1/20 0.48
CASP6 P55212 2/20 0.48
GAA P10253 2/20 0.47
TLR9 Q9NR96 2/20 0.47
PKM P14618 1/20 0.47
SLC6A2 P23975 1/20 0.46
MGLL Q99685 1/20 0.44
NOTUM Q6P988 1/20 0.44
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692980 0.86 HPGD (0.69) HPGDKMT2AMEN1DRD2DRD5
SCHEMBL143970 0.85 HPGD (1.00) HPGDKMT2AMEN1DRD2DRD5
SCHEMBL31422646 0.85 HPGD (1.00) HPGDKMT2AMEN1DRD2DRD5
SCHEMBL13167920 0.85 HPGD (0.53) HPGDKMT2AMEN1DRD2DRD3
SCHEMBL6763292 0.83 HPGD (0.70) HPGDKMT2AMEN1DRD2DRD3
SCHEMBL4463146 0.83 HPGD (0.74) HPGDKMT2AMEN1TNKSCASP6
SCHEMBL6765903 0.83 HPGD (0.74) HPGDKMT2AMEN1TNKSCASP6
SCHEMBL6328308 0.83 HPGD (0.74) HPGDKMT2AMEN1TNKSCASP6
SCHEMBL16456324 0.83 HPGD (0.74) HPGDKMT2AMEN1TNKSCASP6
SCHEMBL16110543 0.80 OPRK1 (0.65) HPGDKMT2AMEN1TNKSOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677368-B2 4-aryl substituted indolinones SUGEN, INC. 2004-01-13 US claimed
US-20030069297-A1 4-aryl substituted indolinones SUGEN, INC. 2003-04-10 US claimed
CN-104109160-A Pyrrolo-N-heterocyclic compound, preparation method and medicinal application thereof SHANGHAI JIESEN PHARMACEUTICAL CHEMISTRY TECHNOLOGY CO LTD 2014-10-22 CN disclosed
US-6861418-B2 4-aryl substituted indolinones SUGEN, INC. (US) 2005-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030069297-A1 4-aryl substituted indolinones CDK5, CAMK4, TNK2 HPGD 1764/4885KMT2A 1573/4885MEN1 4419/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.