SCHEMBL6334591

SCHEMBL6334591

O=C(Cl)c1cn(-c2ccc(Cl)cc2)c(-c2ccccc2Cl)n1

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 0.64
CNR2 P34972 7/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6335073 0.89 CNR1 (0.64) CNR1CNR2
SCHEMBL6429757 0.88 CNR1 (0.62) CNR1CNR2
SCHEMBL4501902 0.86 CNR1 (0.65) CNR1CNR2
SCHEMBL27591168 0.84 CNR1 (0.67) CNR1CNR2
SCHEMBL5336123 0.83 GABRA2 (0.72) CNR1CNR2
SCHEMBL6533838 0.83 GABRA2 (0.72) CNR1CNR2
SCHEMBL5808097 0.82 CNR1 (0.74) CNR1CNR2
SCHEMBL6335983 0.82 CNR1 (0.59) CNR1CNR2
SCHEMBL27591192 0.82 CNR1 (0.57) CNR1CNR2
SCHEMBL27609608 0.82 CNR1 (0.64) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1865248-A Imidazole-4-carboxamide derivatives, preparation and use thereof for treatment of obesity BAYER PHARMACEUTICALS CORP (US) 2006-11-22 CN disclosed
US-20050256167-A1 Preparation and use of imidazole derivatives for treatment of obesity BAYER PHARMACEUTICALS CORPORATION (US) 2005-11-17 US disclosed
US-6960601-B2 Preparation and use of imidazole derivatives for treatment of obesity BAYER PHARMACEUTICALS CORPORATION (US) 2005-11-01 US disclosed
WO-2005099705-A2 PREPARATION OF IMIDAZOLE DERIVATIVES AND METHODS OF USE BAYER PHARMACEUTICALS CORPORATION (US) 2005-10-27 WO disclosed
CN-1599724-A Imidazole-4-carboxamide derivatives, their preparation and use in the treatment of obesity BAYER PHARMACEUTICALS CORPORAT (US) 2005-03-23 CN disclosed
EP-1432691-A1 IMIDAZOLE-4-CARBOXAMIDE DERIVATIVES, PREPARATION AND USE THEREOF FOR TREATMENT OF OBESITY Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
US-20040063691-A1 Preparation and use of imidazole derivatives for treatment of obesity BAYER PHARMACEUTICALS CORPORATION 2004-04-01 US disclosed
WO-2003040107-A1 IMIDAZOLE-4-CARBOXAMIDE DERIVATIVES, PREPARATION AND USE THEREOF FOR TREATMENT OF OBESITY BAYER PHARMACEUTICALS CORPORATION (US) 2003-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063691-A1 Preparation and use of imidazole derivatives for treatment of obesity GPR119, GIPR, PGC CNR1 405/4885CNR2 340/4885
US-20050256167-A1 Preparation and use of imidazole derivatives for treatment of obesity GPR119, GIPR, PGC CNR1 405/4885CNR2 340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.