SCHEMBL6338134

SCHEMBL6338134

COc1ccc2ccn(S(=O)(=O)c3ccc4c(c3)CNCC4(C)C)c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 10/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CYP3A4 P08684 1/20 0.48
FABP4 P15090 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
POLB P06746 1/20 0.44
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
PPARG P37231 2/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6332940 0.86 HTR6 (0.51) HTR6CYP3A4PPARGPPARDPPARA
SCHEMBL6328502 0.83 HTR6 (0.40) HTR6CYP3A4
SCHEMBL6338119 0.82 HTR6 (0.61) HTR6MEN1KMT2ACYP3A4FABP4
SCHEMBL6330490 0.74 HTR6 (0.61) HTR6MEN1KMT2ACYP3A4L3MBTL1
SCHEMBL1892670 0.73 HTR6 (0.78) HTR6MEN1KMT2ACYP3A4FABP4
SCHEMBL29559974 0.72 MEN1 (1.00) HTR6MEN1KMT2ACYP3A4FABP4
SCHEMBL10345778 0.72 MEN1 (1.00) HTR6MEN1KMT2ACYP3A4FABP4
SCHEMBL6331024 0.70 HTR6 (0.52) HTR6FABP4L3MBTL1KDM4E
SCHEMBL3177100 0.68 KCNH2 (0.43) CYP3A4TSHR
SCHEMBL6332254 0.68 PNMT (0.52) HTR6CYP3A4PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849644-B2 Isoquinoline derivatives useful in the treatment of CNS disorders SMITHKLINE BEECHAM P.L.C. (GB) 2005-02-01 US claimed