SCHEMBL6328502

SCHEMBL6328502

CC1(C)CNCc2cc(S(=O)(=O)n3ccc4ccc(C(F)(F)F)cc43)ccc21

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 19/20 0.40
RORC P51449 1/20 0.38
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
CYP3A4 P08684 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6332940 0.85 HTR6 (0.51) HTR6HTR1ADRD2CYP3A4
SCHEMBL6338134 0.83 HTR6 (0.55) HTR6CYP3A4
SCHEMBL6338175 0.82 HTR6 (0.48) HTR6RORCCYP3A4
SCHEMBL6166989 0.79 HTR6 (0.56) HTR6CYP3A4
SCHEMBL12968852 0.75 PNMT (0.42)
SCHEMBL15566251 0.74 ALDH1A1 (0.49) HTR6RORCHTR1ADRD2
SCHEMBL6331024 0.71 HTR6 (0.52) HTR6
SCHEMBL45741 0.71 HTR6 (0.63) HTR6RORCHTR1ADRD2CYP3A4
SCHEMBL31319736 0.71 HTR6 (0.63) HTR6RORCHTR1ADRD2CYP3A4
SCHEMBL6330560 0.68 HTR6 (0.58) HTR6HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849644-B2 Isoquinoline derivatives useful in the treatment of CNS disorders SMITHKLINE BEECHAM P.L.C. (GB) 2005-02-01 US claimed