SCHEMBL633936

SCHEMBL633936

O=C(NC1CCOC1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.61
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
KDM1A O60341 1/20 0.50
HPGDS O60760 1/20 0.49
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
CTSK P43235 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29167802 1.00 NAMPT (0.61) NAMPTNPC1RAB9AMEN1KMT2A
SCHEMBL13868569 1.00 NAMPT (0.61) NAMPTNPC1RAB9AMEN1KMT2A
SCHEMBL364174 0.90 NPC1 (0.62) NAMPTNPC1RAB9AMEN1KMT2A
Water SCHEMBL30838095 0.88 NPC1 (0.60) NAMPTNPC1RAB9AMEN1KMT2A
SCHEMBL12505662 0.86 NPC1 (0.56) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL14797411 0.84 NAMPT (0.52) NAMPTNPC1RAB9AMEN1KMT2A
SCHEMBL27962735 0.83 KDM1A (0.54) NAMPTNPC1RAB9AKDM1AHPGDS
SCHEMBL30968148 0.83 ALDH1A1 (0.52) NAMPTNPC1RAB9AMEN1KMT2A
SCHEMBL30968047 0.83 ALDH1A1 (0.52) NAMPTNPC1RAB9AMEN1KMT2A
SCHEMBL23387883 0.82 ALDH1A1 (0.59) NAMPTRAB9ASMN1; SMN2HPGDSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117647598-A High performance liquid analysis method for enantiomer of (S) -3-amino tetrahydrofuran and intermediate 上海司太立制药有限公司 2024-03-05 CN claimed
EP-1126843-A4 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS THAT ARE INHIBITORS OF IMPDH ENZYME BRISTOL MYERS SQUIBB CO (US) 2005-06-15 EP claimed
EP-1126843-A1 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS THAT ARE INHIBITORS OF IMPDH ENZYME BRISTOL-MYERS SQUIBB COMPANY (US) 2001-08-29 EP claimed
WO-2000025780-A1 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS THAT ARE INHIBITORS OF IMPDH ENZYME BRISTOL-MYERS SQUIBB COMPANY (US) 2000-05-11 WO claimed
EP-4630410-A1 POLQ INHIBITORS Astrazeneca AB (SE) 2025-10-15 EP disclosed
CN-113382730-B Selective glucocorticoid receptor modifier for use in the treatment of impaired skin wound healing 阿克里斯生物医药有限公司 2025-02-25 CN disclosed
CN-115697993-B Pyrimidine compounds as AXL inhibitors 南京正大天晴制药有限公司 2024-12-10 CN disclosed
WO-2024121753-A1 POLQ INHIBITORS ASTRAZENECA AB (SE) 2024-06-13 WO disclosed
CN-117647598-A High performance liquid analysis method for enantiomer of (S) -3-amino tetrahydrofuran and intermediate 上海司太立制药有限公司 2024-03-05 CN disclosed
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
US-20230227484-A1 PYRIMIDINE COMPOUND AS AXL INHIBITOR NANJING CHIA TAI TIANQING PHARMACEUTICAL CO., LTD. (CN) 2023-07-20 US disclosed
CN-111655700-B Oxadiazolopyridine derivatives as ghrelin O-acyltransferase (GOAT) inhibitors 勃林格殷格翰国际有限公司 2023-07-18 CN disclosed
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed
EP-3568390-A1 SMALL MOLECULE ACTIVATORS OF NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE (NAMPT) AND USES THEREOF Sanford Burnham Prebys Medical Discovery Institute (US) 2019-11-20 EP disclosed
US-10421734-B1 Process for the preparation of enantiopure 3-amino tetrahydrofuran and its salts SAMI LABS LIMITED (IN) 2019-09-24 US disclosed
WO-2018132372-A1 SMALL MOLECULE ACTIVATORS OF NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE (NAMPT) AND USES THEREOF Sanford Burnham Prebys Medical Discovery Institute (US) 2018-07-19 WO disclosed
EP-2419423-A1 FLUORO SUBSTITUTED PYRIMIDINE COMPOUNDS AS JAK3 INHIBITORS Cellzome Limited (GB) 2012-02-22 EP disclosed
WO-2010118986-A1 FLUORO SUBSTITUTED PYRIMIDINE COMPOUNDS AS JAK3 INHIBITORS CELLZOME LIMITED (GB) 2010-10-21 WO disclosed
US-7514573-B2 Processes for the manufacture of chiral and racemic forms of 3-aminotetrahydrofurans, their salts and derivatives SAMI LABS LTD (IN) 2009-04-07 US disclosed
US-20080255377-A1 reduction of diesters of aspartic acid, then cyclization with the aid of sulfonic acids, hydrolysis using a base to give 3-(S)-aminotetrahydrofuran as its hydrochloride or p-toluenesulfonate salt, or as base itself MAJEED MUHAMMED 2008-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080255377-A1 reduction of diesters of aspartic acid, then cyclization with the aid of sulfonic acids, hydrolysis using a base to give 3-(S)-aminotetrahydrofuran as its hydrochloride or p-toluenesulfonate salt, or as base itself AASDHPPT, DNPEP, ASNS NAMPT 780/4885NPC1 4777/4885RAB9A 4799/4885
US-20230227484-A1 PYRIMIDINE COMPOUND AS AXL INHIBITOR AXL, FLT3, TYMP NAMPT 43/4885NPC1 4461/4885RAB9A 2614/4885
US-10421734-B1 Process for the preparation of enantiopure 3-amino tetrahydrofuran and its salts AASDHPPT, AAAS, AADAT NAMPT 1017/4885NPC1 4097/4885RAB9A 2239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.