SCHEMBL634716

SCHEMBL634716

CN(C)C(=O)c1cccc2cc(-c3ccc4c(C(N)=O)cccc4c3)ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
GAA P10253 1/20 0.53
ERN1 O75460 3/20 0.45
PARP1 P09874 6/20 0.44
DHODH Q02127 1/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
AURKA O14965 4/20 0.41
MET P08581 4/20 0.41
KDR P35968 4/20 0.41
TEK Q02763 4/20 0.41
AURKB Q96GD4 4/20 0.41
PTPN1 P18031 1/20 0.41
ABL1 P00519 1/20 0.40
LCK P06239 1/20 0.40
LYN P07948 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL634882 0.89 KDM4E (0.65) KDM4EALDH1A1GAAERN1PARP1
SCHEMBL14134468 0.85 PARP1 (0.47) ERN1PARP1DHODHHSD17B1HSD17B2
SCHEMBL14052345 0.81 PARP1 (0.50) ERN1PARP1HSD17B1HSD17B2ABL1
SCHEMBL353489 0.81 ALDH1A1 (0.53) KDM4EALDH1A1GAAERN1PARP1
SCHEMBL31612414 0.78 KDM4E (0.56) KDM4EALDH1A1GAAPARP1MEN1
SCHEMBL355056 0.78 HSD17B1 (0.43) KDM4EALDH1A1GAAPARP1HSD17B1
SCHEMBL353654 0.77 HSD17B2 (0.43) KDM4EALDH1A1GAAPARP1HSD17B1
SCHEMBL10407111 0.77 NR4A1 (0.59) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL353378 0.76 F10 (0.48) KDM4EALDH1A1GAAPARP1MEN1
SCHEMBL355595 0.76 TRPM8 (0.46) KDM4EALDH1A1GAAPARP1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418942-A1 NAPHTHALENE-BASED INHIBITORS OF ANTI-APOPTOTIC PROTEINS Sanford-Burnham Medical Research Institute (US) 2012-02-22 EP disclosed