SCHEMBL6377804

SCHEMBL6377804

O=C(c1ccccc1)c1csc(Br)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.56
ALDH1A1 P00352 2/20 0.54
ATM Q13315 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
ALOX15 P16050 1/20 0.47
HTT P42858 1/20 0.47
SRD5A2 P31213 1/20 0.47
HPGDS O60760 1/20 0.44
PBRM1 Q86U86 1/20 0.44
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
HPGD P15428 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 3/20 0.41
LMNA P02545 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27682287 0.88 CES2 (0.39) CA2ALDH1A1TDP1RAB9ALMNA
SCHEMBL28542772 0.78 CA2 (0.57) CA2ALDH1A1ATMTDP1L3MBTL1
SCHEMBL4110334 0.77 DAO (0.62) CA2ALDH1A1ATMTDP1L3MBTL1
SCHEMBL31287853 0.77 DAO (0.62) CA2ALDH1A1ATMTDP1L3MBTL1
SCHEMBL10367856 0.76 ATM (0.55) CA2ALDH1A1ATMTDP1L3MBTL1
Benzophenone SCHEMBL28127869 0.73 ALDH1A1 (0.88) ALDH1A1ATMTDP1L3MBTL1SRD5A2
Benzophenone SCHEMBL6061130 0.73 ALDH1A1 (1.00) CA2ALDH1A1ATMTDP1L3MBTL1
Benzophenone SCHEMBL30536983 0.73 ALDH1A1 (1.00) CA2ALDH1A1ATMTDP1L3MBTL1
Benzophenone SCHEMBL30537001 0.73 ALDH1A1 (1.00) CA2ALDH1A1ATMTDP1L3MBTL1
Benzophenone SCHEMBL28491203 0.73 ALDH1A1 (1.00) CA2ALDH1A1ATMTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100334085-C Quinuclidine compound and medicine containing the same as active ingredient EISAI R & D CO LTD (JP) 2007-08-29 CN disclosed
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
CN-1377349-A Quinuclidine compound and medicine containing the same as active ingredient EISAI CO LTD (JP) 2002-10-30 CN disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed