SCHEMBL6378374

SCHEMBL6378374

CN(Cc1cc(C(=O)OC(C)(C)C)ccc1[N+](=O)[O-])C(=O)CO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
THRB P10828 4/20 0.39
VCAM1 P19320 1/20 0.38
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
CRHBP P24387 1/20 0.37
RAB9A P51151 1/20 0.37
CRHR2 Q13324 1/20 0.37
POLB P06746 2/20 0.37
LMNA P02545 2/20 0.36
ATM Q13315 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MET P08581 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6655650 0.88 KMT2A (0.43) KMT2AMEN1THRBVCAM1MAPT
SCHEMBL6378830 0.83 CASP6 (0.53) POLBLMNA
SCHEMBL6948552 0.82 KMT2A (0.44) KMT2AMEN1THRBVCAM1MAPT
SCHEMBL7450087 0.81 PDK1 (0.42) KMT2ATHRBVCAM1MAPTALDH1A1
SCHEMBL7613643 0.81 ESR1 (0.49) KMT2AMEN1THRBMAPTALDH1A1
SCHEMBL6378448 0.80 KMT2A (0.44) KMT2AMEN1VCAM1MAPTALDH1A1
SCHEMBL6378524 0.78 VCAM1 (0.43) KMT2AMEN1VCAM1MAPTALDH1A1
SCHEMBL11247732 0.77 CASP6 (0.57) KMT2AVCAM1MAPTALDH1A1NPC1
SCHEMBL8329755 0.76 KMT2A (0.40) KMT2AMEN1THRBVCAM1MAPT
SCHEMBL8326945 0.76 KMT2A (0.40) KMT2AMEN1THRBVCAM1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1225895-B1 FAB I INHIBITORS AFFINIUM PHARM INC (CA) 2005-05-04 EP disclosed
US-6762201-B1 SUCH AS N-((2-AMINO-5-(N-METHYL-N-((1-METHYLINDOL-2-YL) -METHYL)CARBAMOYL)PHENYL)METHYL)-N-METHYLACETAMIDE; BACTERIAL INFECTIONS AFFINIUM PHARMACEUTICALS, INC. (CA) 2004-07-13 US disclosed