SCHEMBL6380847

SCHEMBL6380847

O=C1NC(=O)C(c2cccc3ccccc23)C(=O)N1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.54
KDM1A O60341 1/20 0.50
MTNR1A P48039 1/20 0.46
MAPT P10636 5/20 0.45
ALDH1A1 P00352 5/20 0.45
HPGD P15428 4/20 0.45
NPSR1 Q6W5P4 2/20 0.45
KDM4E B2RXH2 2/20 0.45
TDP2 O95551 1/20 0.45
ALOX12 P18054 1/20 0.45
MAPK1 P28482 1/20 0.45
CASP3 P42574 1/20 0.45
HTT P42858 1/20 0.45
GALK1 P51570 1/20 0.45
BLM P54132 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18025752 0.82 IDO1 (0.51) IDO1KDM1AMTNR1AMAPTALDH1A1
SCHEMBL30588975 0.79 IDO1 (0.55) IDO1KDM1AMTNR1AMAPTALDH1A1
SCHEMBL10822158 0.79 IDO1 (0.55) IDO1KDM1AMTNR1AMAPTALDH1A1
SCHEMBL11876685 0.75 IDO1 (0.37) IDO1MAPTALDH1A1HPGDKDM4E
SCHEMBL9541310 0.74 IDO1 (0.50) IDO1KDM1AMTNR1AMAPTALDH1A1
SCHEMBL23576543 0.74 IDO1 (0.43) IDO1KDM1AMTNR1AMAPTALDH1A1
SCHEMBL9802951 0.73 DDB1 (0.49) ALDH1A1NPSR1KDM4EL3MBTL1TSHR
SCHEMBL6381006 0.73 KDM4E (0.45) IDO1MAPTALDH1A1HPGDKDM4E
SCHEMBL2358320 0.73 MAPT (0.56) IDO1KDM1AMTNR1AMAPTALDH1A1
SCHEMBL24017027 0.73 MTNR1A (0.49) IDO1KDM1AMTNR1AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103370658-B Holographic storage medium and method of making a holographic storage medium 沙特基础全球技术有限公司 2016-08-24 CN disclosed
US-20140212792-A1 HOLOGRAPHIC STORAGE MEDIUM AND METHOD OF MAKING HOLOGRAPHIC STORAGE MEDIUM SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-07-31 US disclosed
US-8728685-B2 Method of making holographic storage medium SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-05-20 US disclosed
EP-2676170-A1 HOLOGRAPHIC STORAGE MEDIUM AND METHOD OF MAKING HOLOGRAPHIC STORAGE MEDIUM SABIC Innovative Plastics IP B.V. (NL) 2013-12-25 EP disclosed
CN-103370658-A Holographic storage medium and method of making a holographic storage medium SABIC INNOVATIVE PLASTICS IP 2013-10-23 CN disclosed
WO-2012138421-A1 HOLOGRAPHIC STORAGE MEDIUM AND METHOD OF MAKING HOLOGRAPHIC STORAGE MEDIUM SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2012-10-11 WO disclosed
US-20120208110-A1 HOLOGRAPHIC STORAGE MEDIUM AND METHOD OF MAKING HOLOGRAPHIC STORAGE MEDIUM SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2012-08-16 US disclosed
CN-1318406-C New barbituric acid derivatives, processes for their prodn. and pharmaceutical agent contg. same BOEHRINGER MANNHEIM GMBH (DE) 2007-05-30 CN disclosed
CN-1295227-C Barbituric acid derivatives with anti-metastatic and anti-tumor activities ROCH DIAGNOSIS EQUIPMENT AG (DE) 2007-01-17 CN disclosed
EP-0989982-B1 BARBITURIC ACID DERIVATIVES WITH ANTIMETASTATIC AND ANTITUMOR ACTIVITY ROCHE DIAGNOSTICS GMBH (DE) 2005-08-17 EP disclosed
US-6472396-B1 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds ROCHE DIAGNOSTICS GMBH (DE) 2002-10-29 US disclosed
EP-0869947-B1 BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2002-10-23 EP disclosed
US-6335332-B1 MATRIX METALLOPROTEASE INHIBITORS; CONTRACEPTIVES, ANTIINFLAMMATORY AGENTS ROCHE DIAGNOSTICS GMBH (DE) 2002-01-01 US disclosed
CN-1267296-A Barbituric acid derivatives with anti-metastatic and anti-tumor activities ROCH DIAGNOSIS EQUIPMENT AG (DE) 2000-09-20 CN disclosed
US-6110924-A MATRIX METALLOPROTEASE INHIBITORS ROCHE DIAGNOSTICS GMBH (DE) 2000-08-29 US disclosed
CN-1209123-A New barbituric acid derivatives, processes for their prodn. and pharmaceutical agent contg. same BOEHRINGER MANNHEIM GMBH (DE) 1999-02-24 CN disclosed
EP-0869947-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1998-10-14 EP disclosed
WO-1997023465-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1997-07-03 WO disclosed