Pyridine

Pyridine

SCHEMBL638445

COC(=O)Cc1ccccc1.c1ccncc1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.56
ALDH1A1 P00352 3/20 0.53
LMNA P02545 2/20 0.53
KDM4E B2RXH2 2/20 0.53
TSHR P16473 1/20 0.51
CYP4F2 P78329 1/20 0.51
CYP4A11 Q02928 1/20 0.51
HPGD P15428 2/20 0.51
RAB9A P51151 3/20 0.51
PKM P14618 2/20 0.51
MAPK1 P28482 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
PAM P19021 1/20 0.49
SLC7A5 Q01650 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 2/20 0.46
HSP90AB1 P08238 1/20 0.46
NFKB1 P19838 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methyl Alcohol SCHEMBL3396251 0.91 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2
SCHEMBL1870609 0.89 ALDH1A1 (0.62) ALDH1A1LMNAKDM4ETSHRCYP4F2
SCHEMBL4675 0.89 ALDH1A1 (0.62) ALDH1A1LMNAKDM4ETSHRCYP4F2
Benzene SCHEMBL28096336 0.89 ALDH1A1 (0.62) ALDH1A1LMNAKDM4ETSHRCYP4F2
Methane SCHEMBL10924043 0.87 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2
Hydrochloric Acid SCHEMBL9268979 0.87 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2
Hydrogen Sulfide SCHEMBL28016697 0.87 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2
Ammonia Solution, Strong SCHEMBL38662792 0.87 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2
Ethane SCHEMBL10923525 0.87 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2
Phosphine SCHEMBL27697952 0.87 ALDH1A1 (0.61) ALDH1A1LMNAKDM4ETSHRCYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506961-B1 Processes for resolving piperidyl acetamide stereoisomers CELGENE CORP (US) 2012-02-22 EP disclosed
EP-1612207-B1 Processes and intermediates for preparing 2-substituted piperidine stereoisomers CELGENE CORP (US) 2009-01-07 EP disclosed
US-7459560-B2 Processes and intermediates for resolving piperidyl acetamide stereoisomers CELGENE CORPORATION (US) 2008-12-02 US disclosed
US-20060142583-A1 Processes and intermediates for resolving piperidyl acetamide stereoisomers KHETANI VIKRAM 2006-06-29 US disclosed
EP-1612207-A1 Processes and intermediates for preparing 2-substituted piperidine stereoisomers CELGENE CORPORATION (US) 2006-01-04 EP disclosed
US-6962997-B1 Process and intermediates for resolving piperidyl acetamide steroisomers CELGENE CORPORATION (US) 2005-11-08 US disclosed
EP-1082307-B1 PROCESSES AND INTERMEDIATES FOR PREPARING 2-SUBSTITUTED PIPERIDINE STEREOISOMERS CELGENE CORP (US) 2005-09-14 EP disclosed
EP-1506961-A2 Processes and intermediates for resolving piperidyl acetamide stereoisomers CELGENE CORPORATION (US) 2005-02-16 EP disclosed
US-20050014790-A1 Processes and intermediates for resolving piperidyl acetamide stereoisomers CELGENE CORPORATION 2005-01-20 US disclosed
EP-0983238-B1 PROCESSES AND INTERMEDIATES FOR RESOLVING PIPERIDYL ACETAMIDE STEREOISOMERS CELGENE CORP (US) 2004-08-18 EP disclosed
US-6359139-B1 REACTING 1-THREO-PIPERIDYL ACETAMIDE WITH AN ALKANOIC ACID IN SOLVNET CELGENE CORPORATION 2002-03-19 US disclosed
EP-0983238-A4 PROCESSES AND INTERMEDIATES FOR RESOLVING PIPERIDYL ACETAMIDE STEREOISOMERS CELGENE CORP (US) 2001-08-08 EP disclosed
EP-0983238-A1 PROCESSES AND INTERMEDIATES FOR RESOLVING PIPERIDYL ACETAMIDE STEREOISOMERS CELGENE CORPORATION (US) 2000-03-08 EP disclosed
US-5965734-A REACTING 2-SUBSTITUTED PYRIDINE WITH HYDROGEN IN THE PRESENCE OF CATALYST AND ALKANOIC ACID, ADDING AKLYL ALKANOATE, AND THEN REACTING WITH AQUEOUS BASE THEN WITH ACID AND RESOLVING AGENT TO FORM ACID SALTS OF 1-ERYTHRO PIPERIDINE STEREOSIOMERS CELGENE CORPORATION (US) 1999-10-12 US disclosed
US-5936091-A Processes and intermediates for resolving piperidyl acetamide stereoisomers CELGENE CORPORATION (US) 1999-08-10 US disclosed
WO-1998052921-A1 PROCESSES AND INTERMEDIATES FOR RESOLVING PIPERIDYL ACETAMIDE STEREOISOMERS CELGENE CORPORATION (US) 1998-11-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014790-A1 Processes and intermediates for resolving piperidyl acetamide stereoisomers NAAA, DHPS, CTPS2 CYP19A1 1729/4885ALDH1A1 321/4885LMNA 2492/4885
US-20060142583-A1 Processes and intermediates for resolving piperidyl acetamide stereoisomers NAAA, DHPS, CTPS2 CYP19A1 1729/4885ALDH1A1 321/4885LMNA 2492/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.