SCHEMBL6399178

SCHEMBL6399178

COc1cccc(C(=O)CN2C=CN(CC(=O)c3cccc(F)c3)C2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
GRIN2B Q13224 2/20 0.59
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
CDYL2 Q8N8U2 5/20 0.54
CDYL Q9Y232 5/20 0.54
CBX7 O95931 3/20 0.54
SMN1; SMN2 Q16637 4/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 3/20 0.47
MEN1 O00255 1/20 0.47
CDY1; CDY1B Q9Y6F8 4/20 0.47
MAPT P10636 2/20 0.47
HPGD P15428 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
CHRM3 P20309 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722012 0.88 GRIN2B (0.52) GRIN2BNPC1RAB9ASMN1; SMN2KMT2A
Bromide SCHEMBL6074281 0.85 NPC1 (0.49) ALDH1A1GRIN2BNPC1RAB9ACDYL2
SCHEMBL10531109 0.85 MAPT (0.51) ALDH1A1GRIN2BNPC1RAB9ACDYL2
SCHEMBL6401176 0.84 GRIN2B (0.55) GRIN2BNPC1SMN1; SMN2KMT2AKDM4E
Hydrochloric Acid SCHEMBL10528594 0.84 MAPT (0.50) ALDH1A1GRIN2BNPC1RAB9ACDYL2
Bromide SCHEMBL3853590 0.84 NPC1 (0.53) ALDH1A1GRIN2BNPC1RAB9ACDYL2
Iodide SCHEMBL10531088 0.84 MAPT (0.50) ALDH1A1GRIN2BNPC1RAB9ACDYL2
Bromide SCHEMBL10526720 0.84 NPC1 (0.53) ALDH1A1GRIN2BNPC1RAB9ACDYL2
SCHEMBL6399172 0.84 RAB9A (0.58) ALDH1A1GRIN2BNPC1RAB9ACDYL2
SCHEMBL29794014 0.81 CDYL2 (0.46) ALDH1A1GRIN2BNPC1RAB9ACDYL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272936-A1 Imidazolium cxcr3 inhibitors SMITHKLINE BEECHAM CORPORATION 2005-12-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050272936-A1 Imidazolium cxcr3 inhibitors CXCR3, CXCR1, CCR7 ALDH1A1 1784/4885GRIN2B 1128/4885NPC1 1098/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.