SCHEMBL6399255

SCHEMBL6399255

CCc1ccc(Nc2c(-c3nnc(N(C)CC4CCCCO4)o3)ccc(F)c2F)c(F)c1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.31
LMNA P02545 2/20 0.31
CSF1R P07333 1/20 0.31
TRPC5 Q9UL62 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204476 0.87 PDE8B (0.32) TRPC5
SCHEMBL6207134 0.84 TUBB4A (0.37) CNR2LMNATRPC5
SCHEMBL6399021 0.79 CRHR1 (0.33) CNR2LMNA
SCHEMBL6281375 0.78 IDO1 (0.33)
SCHEMBL6400380 0.78 FLT1 (0.32)
SCHEMBL6207240 0.78
SCHEMBL6206842 0.77
SCHEMBL6207023 0.77 HTR2A (0.31)
SCHEMBL6206400 0.76
SCHEMBL6400419 0.75 KDM4E (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050004186-A1 MEK inhibiting compounds PFIZER INC 2005-01-06 US claimed
US-20050004186-A1 MEK inhibiting compounds PFIZER INC 2005-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004186-A1 MEK inhibiting compounds MAPK1, MAP3K1, MAPK3 CNR2 1401/4885LMNA 3833/4885CSF1R 507/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.