SCHEMBL6399738

SCHEMBL6399738

Cc1cccc(C#Cc2ccc3c(c2)N(CCN2CCOCC2)C(=O)CO3)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.48
CYP2C19 P33261 4/20 0.48
CYP3A4 P08684 3/20 0.48
GRM5 P41594 2/20 0.45
HTR1A P08908 7/20 0.43
HTR1D P28221 7/20 0.43
HTR1B P28222 7/20 0.43
SLC6A4 P31645 1/20 0.43
EGFR P00533 7/20 0.43
RIPK1 Q13546 1/20 0.42
KCNH2 Q12809 1/20 0.42
CYP1A2 P05177 4/20 0.41
CYP2D6 P10635 2/20 0.41
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6393258 0.88 HTT (0.47) CYP2C9CYP2C19CYP3A4GRM5HTR1A
SCHEMBL6393501 0.86 RIPK1 (0.42) CYP2C9CYP2C19CYP3A4GRM5HTR1A
SCHEMBL6391869 0.85 HTR1A (0.47) CYP2C9CYP2C19CYP3A4GRM5HTR1A
SCHEMBL6392491 0.85 RIPK1 (0.42) CYP2C9CYP2C19CYP3A4GRM5HTR1A
SCHEMBL6393526 0.85 REN (0.45) CYP2C9CYP2C19CYP3A4GRM5HTR1A
SCHEMBL6178668 0.82 RIPK1 (0.47) CYP2C9CYP2C19CYP3A4GRM5HTR1A
SCHEMBL6395028 0.77 GRM5 (0.50) CYP2C9CYP2C19CYP3A4GRM5RIPK1
SCHEMBL23076327 0.76 RIPK1 (0.48) CYP2C9CYP2C19CYP3A4GRM5RIPK1
SCHEMBL6426996 0.76 GRM5 (0.44) CYP2C9CYP2C19CYP3A4GRM5RIPK1
SCHEMBL6168702 0.73 HTT (0.45) CYP2C9CYP2C19CYP3A4HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050165011-A1 Benzoxazine and benzoxazinone substituted triazoles GELLIBERT FRANCOISE J (FR) 2005-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165011-A1 Benzoxazine and benzoxazinone substituted triazoles ACVR1, TGFBR1, SMAD3 CYP2C9 3071/4885CYP2C19 2960/4885CYP3A4 1867/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.