SCHEMBL6402495

SCHEMBL6402495

Cc1ccccc1C(=O)NCc1cc(C(=O)Nc2ccccc2)no1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.56
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
POLB P06746 1/20 0.49
MAPK1 P28482 3/20 0.48
KCNK3 O14649 1/20 0.48
KCNK9 Q9NPC2 1/20 0.48
TYK2 P29597 1/20 0.48
MAPT P10636 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
FFAR1 O14842 1/20 0.47
PPARG P37231 1/20 0.47
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6402278 0.84 HDAC6 (0.57) SMN1; SMN2NPC1RAB9APOLBMAPK1
SCHEMBL6410519 0.83 NPC1 (0.59) HPGDSMN1; SMN2NPC1RAB9APOLB
SCHEMBL6402219 0.81 POLB (0.55) SMN1; SMN2NPC1RAB9APOLBMAPK1
SCHEMBL6410595 0.81 HPGD (0.51) HPGDSMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL6403903 0.80 PPARG (0.55) SMN1; SMN2NPC1RAB9APOLBMAPK1
SCHEMBL6408049 0.78 NPC1 (0.55) HPGDSMN1; SMN2NPC1RAB9APOLB
SCHEMBL21993 0.74 HPGD (1.00) HPGDSMN1; SMN2NPC1RAB9APOLB
SCHEMBL8266868 0.73 RAB9A (0.77) SMN1; SMN2NPC1RAB9AMAPTCYP1A2
SCHEMBL6408618 0.71 SMN1; SMN2 (0.62) HPGDSMN1; SMN2NPC1RAB9APOLB
Iodomethane SCHEMBL20530190 0.71 HPGD (0.93) HPGDSMN1; SMN2NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528737-B Novel heteroaryl carboxamides HOFFMANN LA ROCHE 2012-07-04 CN disclosed
US-20050171358-A1 Substituted isoxazole alkylamine derivative and agri-and horticultural fungicide SDS BIOTECH K.K. (JP) 2005-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171358-A1 Substituted isoxazole alkylamine derivative and agri-and horticultural fungicide AHR, ERG28, CYP1A2 HPGD 3244/4885SMN1; SMN2 4458/4885NPC1 1915/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.