SCHEMBL6412015

SCHEMBL6412015

Cc1cnc(C(=O)N2CCN(C(=O)C3=NOC4(CCN(S(=O)(=O)c5ccc(F)cc5)CC4)C3)CC2)cn1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
GAA P10253 2/20 0.48
PKM P14618 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
LMNA P02545 1/20 0.40
GPR183 P32249 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2402487 0.79 KDM4E (0.50) ALDH1A1GAAL3MBTL1LMNA
SCHEMBL6409630 0.78 ALDH1A1 (0.48) ALDH1A1GAAPKML3MBTL1LMNA
SCHEMBL2399286 0.77 TGM2 (0.49) ALDH1A1GAAPKM
SCHEMBL2581274 0.76 F13A1 (0.46) ALDH1A1GAAPKMLMNA
SCHEMBL6415538 0.74 ALDH1A1 (0.44) ALDH1A1GAAPKML3MBTL1LMNA
SCHEMBL6411306 0.74 LMNA (0.51) ALDH1A1GAALMNA
SCHEMBL2400362 0.73 GAA (0.65) ALDH1A1GAAPKML3MBTL1LMNA
SCHEMBL6410715 0.73 LMNA (0.46) ALDH1A1GAAPKML3MBTL1LMNA
SCHEMBL6416697 0.72 CYP2C19 (0.52) ALDH1A1GAAPKML3MBTL1
SCHEMBL6410874 0.72 PKM (0.46) ALDH1A1GAAPKML3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP claimed
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP disclosed
EP-1401841-A1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN Grünenthal GmbH (DE) 2004-03-31 EP disclosed
WO-2003000699-A1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO[4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN Grünenthal GmbH (DE) 2003-01-03 WO disclosed