SCHEMBL641390

SCHEMBL641390

Nc1ccccc1Oc1ccc(Cl)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.63
ALDH1A1 P00352 3/20 0.63
CYP1A2 P05177 2/20 0.63
CYP2C9 P11712 2/20 0.63
CYP2C19 P33261 2/20 0.63
KDM4E B2RXH2 2/20 0.63
MEN1 O00255 1/20 0.63
CYP2D6 P10635 1/20 0.63
HPGD P15428 1/20 0.63
KMT2A Q03164 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
CYP3A4 P08684 1/20 0.61
GAA P10253 2/20 0.58
RCE1 Q9Y256 1/20 0.58
IKBKB O14920 2/20 0.54
HTT P42858 2/20 0.54
LMNA P02545 1/20 0.54
BRAF P15056 1/20 0.54
MAOA P21397 1/20 0.54
MAOB P27338 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29957616 1.00 MAPT (0.63) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL2285909 0.89 GAA (0.69) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL1271606 0.87 GAA (0.67) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6289248 0.87 GAA (0.67) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL1270588 0.87 GAA (0.67) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6289955 0.87 GAA (0.67) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6293151 0.85 GAA (0.64) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6289853 0.85 GAA (0.64) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6290392 0.85 GAA (0.64) MAPTALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL1269990 0.85 GAA (0.64) MAPTALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068437-A Process for producing 2-(p-chlorophenoxy) aniline AMERICAN CYANAMID COMPANY (US) 1991-11-26 US claimed
EP-2950793-B1 COMPOSITION FOR TREATMENT OF PATHOGENS THAT ARE RESISTANT TO TETRACYCLINES BioVersys AG (CH) 2020-04-01 EP disclosed
EP-3551628-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2019-10-16 EP disclosed
US-20190161471-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS INC (US) 2019-05-30 US disclosed
US-10202362-B2 Inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2019-02-12 US disclosed
US-20180162836-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2018-06-14 US disclosed
WO-2018107153-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2018-06-14 WO disclosed
US-9682079-B2 Composition for treatment of pathogens that are resistant to tetracyclines BioVersys AG (CH) 2017-06-20 US disclosed
US-9682079-B2 Composition for treatment of pathogens that are resistant to tetracyclines BioVersys AG (CH) 2017-06-20 US disclosed
US-9682079-B2 Composition for treatment of pathogens that are resistant to tetracyclines BioVersys AG (CH) 2017-06-20 US disclosed
WO-2004002481-A1 ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS NOVO NORDISK A/S (DK) 2004-01-08 WO disclosed
EP-0633145-B1 Thermal recording sheet JUJO PAPER CO LTD (JP) 1998-04-15 EP disclosed
US-5470816-A Urea developers NIPPON PAPER INDUSTRIES CO., LTD. (JP) 1995-11-28 US disclosed
EP-0482508-B1 Biscationic azo dyes and their intermediates BASF AG (DE) 1995-07-12 EP disclosed
US-5424404-A Colorfastness, discoloration inhibition, red and yellow color; coloring paper, leather, printing on polymeric material BASF AKTIENGESELLSCHAFT (DE) 1995-06-13 US disclosed
EP-0633145-A1 Thermal recording sheet NIPPON PAPER INDUSTRIES CO., LTD. (JP) 1995-01-11 EP disclosed
EP-0482508-A1 Biscationic azo dyes and their intermediates BASF Aktiengesellschaft (DE) 1992-04-29 EP disclosed
US-5068437-A Process for producing 2-(p-chlorophenoxy) aniline AMERICAN CYANAMID COMPANY (US) 1991-11-26 US disclosed
US-5068437-A Process for producing 2-(p-chlorophenoxy) aniline AMERICAN CYANAMID COMPANY (US) 1991-11-26 US disclosed
US-4136033-A DIAZO COUPLERS SANDOZ LTD. (CH) 1979-01-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190161471-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE LTA4H, LTC4S, LTB4R MAPT 4121/4885ALDH1A1 1041/4885CYP1A2 241/4885
US-20180162836-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE LTA4H, LTC4S, LTB4R MAPT 4121/4885ALDH1A1 1041/4885CYP1A2 241/4885
US-10202362-B2 Inhibitors of leukotriene A4 hydrolase LTA4H, LTC4S, LTB4R MAPT 4121/4885ALDH1A1 1041/4885CYP1A2 241/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.