SCHEMBL6418671

SCHEMBL6418671

CC(=O)N(C)CC(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.50
TDP1 Q9NUW8 1/20 0.45
HPGD P15428 2/20 0.42
TACR1 P25103 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
MME P08473 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6413830 0.82 AOC3 (0.50) AOC3TACR1ALDH1A1SMN1; SMN2MEN1
SCHEMBL6414328 0.78 TDP1 (0.40) AOC3TDP1HPGDTACR1ALDH1A1
SCHEMBL6414332 0.78 TDP1 (0.40) AOC3TDP1HPGDTACR1ALDH1A1
SCHEMBL6412517 0.74 LMNA (0.40) AOC3TDP1HPGDALDH1A1SMN1; SMN2
SCHEMBL10439829 0.73 HPGD (0.54) HPGDHDAC6ALDH1A1SMN1; SMN2NPSR1
SCHEMBL6411789 0.72 KMT2A (0.45) AOC3TDP1HDAC6ALDH1A1SMN1; SMN2
SCHEMBL2760548 0.72 RIPK1 (0.60) TDP1HDAC6ALDH1A1SMN1; SMN2MAPT
SCHEMBL7496510 0.71 OPRM1 (0.43) AOC3TDP1HPGDHDAC6ALDH1A1
SCHEMBL6413101 0.70 HCRTR1 (0.43) AOC3TDP1HDAC6ALDH1A1KMT2A
SCHEMBL18945572 0.70 HCRTR1 (0.43) AOC3TDP1HDAC6ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050043370-A1 HIV integrase inhibitors WALKER MICHAEL A (US) 2005-02-24 US disclosed
US-6803378-B2 FOR THERAPY AND PROPHYLAXIS OF ACQUIRED IMMUNE DEFICIENCY SYNDROME (AIDS), OR ARC BRISTOL-MYERS SQUIBB COMPANY 2004-10-12 US disclosed
US-20030181490-A1 HIV integrase inhibitors WALKER MICHAEL A (US) 2003-09-25 US disclosed
US-20030027847-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2003-02-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043370-A1 HIV integrase inhibitors AKR1C3, CBR3, CBR1 AOC3 66/4885TDP1 1762/4885HPGD 592/4885
US-20030181490-A1 HIV integrase inhibitors CBR1, CCR5, CCR1 AOC3 124/4885TDP1 863/4885HPGD 1410/4885
US-20030027847-A1 HIV integrase inhibitors CBR1, CCR5, CCR1 AOC3 124/4885TDP1 863/4885HPGD 1410/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.