SCHEMBL6419873

SCHEMBL6419873

CC(C)(CO)NC(=O)c1ccccc1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
NPC1 O15118 5/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 1/20 0.49
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
RAB9A P51151 4/20 0.47
ATM Q13315 1/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL28774251 0.98 GAA (0.59) GAAMEN1KMT2ATDP1NPC1
SCHEMBL8465283 0.87 CES2 (0.49) GAAKMT2ANPC1HPGDRAB9A
SCHEMBL10330517 0.87 NPSR1 (0.58) GAAMEN1KMT2ATDP1NPC1
SCHEMBL6420811 0.82 GAA (0.63) GAAMEN1KMT2ATDP1NPC1
SCHEMBL2886082 0.81 KMT2A (0.49) GAAMEN1KMT2ANPC1MAPT
SCHEMBL6419790 0.81 CNR2 (0.51) NPC1RAB9AATMCES2CES1
SCHEMBL6419694 0.81 CNR2 (0.54) GAANPC1SMN1; SMN2RAB9AATM
SCHEMBL11838628 0.80 RAB9A (0.48) MEN1KMT2ANPC1ALDH1A1MAPT
SCHEMBL27413434 0.80 POLB (0.55) KMT2ANPC1ALDH1A1MAPTHPGD
SCHEMBL6421030 0.80 ACVR1B (0.50) NPC1ALDH1A1HPGDSMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1034783-B1 AMIDE DERIVATIVES FOR THE TREATMENT OF RETINAL NEURODEGENERATIVE DISORDERS SUMITOMO PHARMA (JP) 2004-12-15 EP claimed
US-20020147204-A1 Amide derivative SUMITOMO PHARMACEUTICALS COMPANY, LIMITED 2002-10-10 US claimed
CN-1278167-A Amide derivatives SUMITOMO PHARMA (JP) 2000-12-27 CN claimed
EP-1034783-A1 AMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP claimed
CN-1856304-A Heteroaromatic ureas that modulate the function of the capsaicin-1 receptor (VR1) MERCK SHARP & DOHME (GB) 2006-11-01 CN disclosed
US-6936736-B2 Amide derivative SUMITOMO MANUFACTURING COMPANY LIMITED (JP) 2005-08-30 US disclosed
EP-1034783-B1 AMIDE DERIVATIVES FOR THE TREATMENT OF RETINAL NEURODEGENERATIVE DISORDERS SUMITOMO PHARMA (JP) 2004-12-15 EP disclosed
US-20020147204-A1 Amide derivative SUMITOMO PHARMACEUTICALS COMPANY, LIMITED 2002-10-10 US disclosed
US-6384033-B1 DRUGS FOR VISION DEFECTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2002-05-07 US disclosed
EP-1184367-A1 AMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2002-03-06 EP disclosed
CN-1278167-A Amide derivatives SUMITOMO PHARMA (JP) 2000-12-27 CN disclosed
EP-1034783-A1 AMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP disclosed
CN-1218472-A Pharmaceutically useful compounds ASTRA PHARMA PROD (GB) 1999-06-02 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020147204-A1 Amide derivative ALDH1A2, NR1H2, HDAC3 GAA 3670/4885MEN1 3899/4885KMT2A 1003/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.