SCHEMBL6423002

SCHEMBL6423002

CC(C(=O)O)N1CCN(C=O)CCN2CCN(CC1)C2=O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GAA P10253 1/20 0.35
HSD17B10 Q99714 1/20 0.33
KCNH2 Q12809 4/20 0.33
HRH3 Q9Y5N1 4/20 0.33
SLC6A9 P48067 1/20 0.32
KMT2A Q03164 3/20 0.32
KDM4E B2RXH2 2/20 0.32
ATM Q13315 1/20 0.31
MEN1 O00255 1/20 0.31
HDAC4 P56524 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423403 0.88 GAA (0.37) ALDH1A1GAASLC6A9KMT2AKDM4E
SCHEMBL6421089 0.80 HSD17B10 (0.34) TSHRALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL2909450 0.77 SIGMAR1 (0.36) TSHRALDH1A1GAAHSD17B10SLC6A9
SCHEMBL24220960 0.74 SLC6A9 (0.40) ALDH1A1CYP1A2CYP2D6KCNH2HRH3
SCHEMBL1133814 0.74
SCHEMBL14100030 0.74 SLC6A9 (0.40) ALDH1A1CYP1A2CYP2D6KCNH2HRH3
SCHEMBL3967181 0.74 SLC6A9 (0.40) ALDH1A1CYP1A2CYP2D6KCNH2HRH3
SCHEMBL7744888 0.74 SLC6A9 (0.40) ALDH1A1CYP1A2CYP2D6KCNH2HRH3
SCHEMBL13223389 0.74 SLC6A9 (0.40) ALDH1A1CYP1A2CYP2D6KCNH2HRH3
SCHEMBL1165366 0.74 SLC6A9 (0.40) ALDH1A1CYP1A2CYP2D6KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047677-B1 Process for the preparation of derivatives of 1,4,7,10-tetraazacyclododecane-1,4-diacetic acid BRACCO SPA (IT) 2005-07-20 EP claimed
EP-1047677-B1 Process for the preparation of derivatives of 1,4,7,10-tetraazacyclododecane-1,4-diacetic acid BRACCO SPA (IT) 2005-07-20 EP disclosed
US-6342597-B1 CONDENSATION REACTION TRIETHYLENETETRAMINE WITH GLYOXAL TO CYCLIZE; OXIDATION, ALKYLATION, HYDROLYSIS, QUATERNIZATION; NUCLEAR MAGNETIC RESONANCE IMAGING DIBRA S.P.A. (IT) 2002-01-29 US disclosed