SCHEMBL6421089

SCHEMBL6421089

CCC(C(=O)O)N1CCN(C=O)CCN2CCN(CC1)C2=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A3 Q01959 2/20 0.33
LMNA P02545 2/20 0.33
SLC6A4 P31645 1/20 0.33
TSHR P16473 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA7 P43166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6422005 0.89 SLC6A2 (0.38) HSD17B10ALDH1A1SLC6A2SLC6A3LMNA
SCHEMBL6422009 0.81 LMNA (0.57) HSD17B10ALDH1A1CYP2C9CYP2C19LMNA
SCHEMBL6423002 0.80 TSHR (0.40) HSD17B10ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL2910332 0.79 OPRD1 (0.38) HSD17B10ALDH1A1CYP2C9SLC6A2SLC6A3
SCHEMBL3102765 0.77
SCHEMBL1462833 0.71 LMNA (0.42) HSD17B10ALDH1A1SLC6A2SLC6A3LMNA
SCHEMBL2909901 0.70 HSD17B10 (0.39) HSD17B10ALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL5617609 0.70 MAPT (0.44) ALDH1A1CYP1A2SLC6A2SLC6A3LMNA
SCHEMBL6420408 0.70 LMNA (0.66) HSD17B10ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11213937 0.70 AR (0.49) HSD17B10ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047677-B1 Process for the preparation of derivatives of 1,4,7,10-tetraazacyclododecane-1,4-diacetic acid BRACCO SPA (IT) 2005-07-20 EP claimed
EP-1047677-B1 Process for the preparation of derivatives of 1,4,7,10-tetraazacyclododecane-1,4-diacetic acid BRACCO SPA (IT) 2005-07-20 EP disclosed
US-6342597-B1 CONDENSATION REACTION TRIETHYLENETETRAMINE WITH GLYOXAL TO CYCLIZE; OXIDATION, ALKYLATION, HYDROLYSIS, QUATERNIZATION; NUCLEAR MAGNETIC RESONANCE IMAGING DIBRA S.P.A. (IT) 2002-01-29 US disclosed