SCHEMBL6426262

SCHEMBL6426262

Cc1cc(C#Cc2ccc(C(C)C(=O)O)cc2)ccc1C1(OC(C)C)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 7/20 0.38
RARG P13631 6/20 0.38
RARA P10276 5/20 0.38
CYP26A1 O43174 1/20 0.38
CYP3A4 P08684 1/20 0.38
CRABP2 P29373 1/20 0.38
AKR1C3 P42330 6/20 0.36
AKR1C2 P52895 5/20 0.36
PTGS2 P35354 8/20 0.35
ACACB O00763 2/20 0.34
PTGS1 P23219 6/20 0.33
LMNA P02545 2/20 0.33
CYP2C9 P11712 2/20 0.33
SLC22A6 Q4U2R8 2/20 0.33
CXCR1 P25024 2/20 0.33
CXCR2 P25025 2/20 0.33
TSHR P16473 2/20 0.33
FFAR1 O14842 1/20 0.33
ALB P02768 1/20 0.33
ESR1 P03372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6425787 0.86 AKR1C3 (0.41) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5736750 0.86 RARB (0.54) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6426294 0.84 RARB (0.37) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6425926 0.83 ACACB (0.42) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5737765 0.83 FFAR1 (0.45) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6426243 0.83 PTGS2 (0.40) RARBAKR1C3AKR1C2PTGS2ACACB
SCHEMBL5735777 0.80 RARA (0.43) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7982072 0.79 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6426280 0.74 PTGS2 (0.41) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6426272 0.74 PTGS2 (0.41) RARBAKR1C3AKR1C2PTGS2ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed