SCHEMBL6426280

SCHEMBL6426280

CCOC1(c2ccc(C#Cc3ccc(C(C)C(=O)O)cc3)cc2C(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.41
ACACB O00763 15/20 0.40
AKR1C3 P42330 2/20 0.39
AKR1C2 P52895 2/20 0.39
RARA P10276 2/20 0.36
RARB P10826 2/20 0.36
RARG P13631 2/20 0.36
CYP26A1 O43174 1/20 0.36
CYP3A4 P08684 1/20 0.36
CRABP2 P29373 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5738841 0.87 RARB (0.51) RARARARBRARGCYP26A1CYP3A4
SCHEMBL6426054 0.85 PTGS2 (0.37) PTGS2ACACBAKR1C3AKR1C2RARA
SCHEMBL5738571 0.85 FFAR1 (0.43) ACACBRARARARBRARGCYP26A1
SCHEMBL5735261 0.83 RARA (0.42) ACACBRARARARBRARGCYP26A1
SCHEMBL7984067 0.82 RARB (0.36) ACACBRARARARBRARGCYP26A1
SCHEMBL7548508 0.81 ACACB (0.34) ACACB
SCHEMBL6425907 0.79 ACACB (0.41) PTGS2ACACBAKR1C3AKR1C2RARA
SCHEMBL6426325 0.78 ACACB (0.38) PTGS2ACACBAKR1C3AKR1C2RARA
SCHEMBL6425926 0.78 ACACB (0.42) PTGS2ACACBAKR1C3AKR1C2RARA
SCHEMBL5738727 0.77 GABRA1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed