SCHEMBL6426703

SCHEMBL6426703

O=C1C(c2ccc(Cl)cc2)=C(C(F)(F)F)C(=O)N1Cc1ccc(F)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
CHRM5 P08912 3/20 0.38
AR P10275 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
TNF P01375 1/20 0.35
CHRM3 P20309 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
CES2 O00748 1/20 0.35
BCHE P06276 1/20 0.35
CES1 P23141 1/20 0.35
CNR1 P21554 2/20 0.34
CNR2 P34972 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
P2RX3 P56373 1/20 0.34
APAF1 O14727 1/20 0.34
CLTC Q00610 1/20 0.34
KCNN4 O15554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427122 0.91 NR1H2 (0.47) NR1H2NR1H3CHRM5CHRM3ALDH1A1
SCHEMBL6426786 0.88 MAPT (0.46) NR1H2NR1H3CHRM5ALDH1A1HTT
SCHEMBL6427820 0.85 KMT2A (0.47) NR1H2NR1H3ALDH1A1HTTMAPT
SCHEMBL6428548 0.84 NR1H2 (0.56) NR1H2NR1H3ALDH1A1CES2BCHE
SCHEMBL6430888 0.82 PKM (0.52) CHRM5ALDH1A1HTTMAPT
SCHEMBL6463014 0.79 CMA1 (0.51) NR1H2NR1H3CHRM5ALDH1A1HTT
SCHEMBL6428843 0.72 NR1H2 (0.52) NR1H2NR1H3ALDH1A1CES2BCHE
SCHEMBL6426845 0.72 MAPT (0.50) NR1H2NR1H3ALDH1A1HTTCES2
SCHEMBL12784743 0.71 CNR1 (0.42) PTGDR2TNFALDH1A1HTTCNR1
SCHEMBL14464973 0.71 CNR1 (0.42) PTGDR2TNFALDH1A1HTTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005024755-A2 MEDICAMENTS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS OR DIABETES DECIPHERA PHARMACEUTICALS, LLC. (US) 2005-03-17 WO disclosed