SCHEMBL6427673

SCHEMBL6427673

Cn1ncc(NC(=O)N2CCC(OC(N)=O)C2)c1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 1/20 0.36
CHRM3 P20309 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 1/20 0.35
NAMPT P43490 1/20 0.35
NPC1 O15118 2/20 0.34
TP53 P04637 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
PDE4B Q07343 1/20 0.33
PI4KB Q9UBF8 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6425495 1.00 ALDH1A1 (0.36) ALDH1A1CYP1A2CHRM3KDM4EHSD17B10
SCHEMBL5497058 0.83 HDAC1 (0.39) ALDH1A1KDM4EHSD17B10NPC1TP53
SCHEMBL5499584 0.83 HDAC1 (0.39) ALDH1A1KDM4EHSD17B10NPC1TP53
SCHEMBL5496605 0.83 HDAC1 (0.39) ALDH1A1KDM4EHSD17B10NPC1TP53
SCHEMBL6430072 0.81 CFD (0.33) CHRM3
SCHEMBL27620821 0.80 HDAC3 (0.49) NAMPT
SCHEMBL6430075 0.80 HDAC3 (0.49) NAMPT
SCHEMBL27620834 0.80 RORC (0.36) CHRM3KDM4ECHRM4CHRM5CHRM1
SCHEMBL5493793 0.80 KDM4E (0.42) ALDH1A1KDM4EHSD17B10TP53SMN1; SMN2
SCHEMBL5493363 0.79 MAPT (0.44) KDM4ENAMPTNPC1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556389-A1 CEPHEM COMPOUNDS Astellas Pharma Inc. (JP) 2005-07-27 EP disclosed
EP-1539164-A1 2-HYDROXY-6-PHENYLPHENANTHRIDINES AS PDE-4 INHIBITORS ALTANA Pharma AG (DE) 2005-06-15 EP disclosed
WO-2004039814-A1 CEPHEM COMPOUNDS ASTELLAS PHARMA INC. (JP) 2004-05-13 WO disclosed
WO-2004019944-A1 2-HYDROXY-6-PHENYLPHENANTHRIDINES AS PDE-4 INHIBITORS ALTANA PHARMA AG (DE) 2004-03-11 WO disclosed