SCHEMBL6428716

SCHEMBL6428716

CCc1cc(C=C(c2ccc3c(c2)C(C)(C)CCC3(C)C)[Si](C)(C)C)sc1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 15/20 0.48
RARG P13631 14/20 0.48
RARA P10276 12/20 0.48
RARB P10826 12/20 0.48
RXRB P28702 9/20 0.48
RXRG P48443 8/20 0.48
CYP26A1 O43174 2/20 0.45
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
GMNN O75496 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
NFKB1 P19838 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427532 0.85 RXRA (0.48) RXRARARGRARARARBRXRB
SCHEMBL177719 0.81 RXRA (0.73) RXRARARGRARARARBRXRB
SCHEMBL177720 0.81 RXRA (0.73) RXRARARGRARARARBRXRB
SCHEMBL6428636 0.78 RARG (0.54) RXRARARGRARARARBRXRB
SCHEMBL6258868 0.76 RARB (0.70) RXRARARGRARARARBRXRB
SCHEMBL6258870 0.76 RARB (0.70) RXRARARGRARARARBRXRB
SCHEMBL6259440 0.76 RXRA (0.48) RXRARARGRARARARBRXRB
SCHEMBL6259442 0.76 RXRA (0.48) RXRARARGRARARARBRXRB
SCHEMBL6428704 0.76 RARB (0.54) RXRARARGRARARARBRXRB
SCHEMBL6428631 0.71 RARA (0.53) RXRARARGRARARARBRXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6906057-B1 Methods for modulating FXR receptor activity ALLERGAN, INC. (US) 2005-06-14 US disclosed