SCHEMBL6429351

SCHEMBL6429351

O=C=CC(Nc1ccc([N+](=O)[O-])cc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
MMP2 P08253 1/20 0.48
MMP9 P14780 1/20 0.48
MMP8 P22894 1/20 0.48
MMP14 P50281 1/20 0.48
MEN1 O00255 7/20 0.46
KMT2A Q03164 7/20 0.46
HPGD P15428 1/20 0.46
ALOX12 P18054 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TGM2 P21980 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 3/20 0.43
MAPT P10636 3/20 0.43
POLB P06746 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6269658 0.82 TGM2 (0.54) CA12CA1MMP2MMP9MMP8
SCHEMBL6429045 0.78 MMP2 (0.42) CA12MMP2MMP9MEN1KMT2A
SCHEMBL14935791 0.73 CA12 (0.54) CA12CA1MMP2MMP9MMP8
SCHEMBL2034750 0.73 CA12 (0.54) CA12CA1MMP2MMP9MMP8
SCHEMBL515914 0.73 CA12 (0.54) CA12CA1MMP2MMP9MMP8
SCHEMBL515915 0.73 CA12 (0.54) CA12CA1MMP2MMP9MMP8
SCHEMBL8373371 0.73 CA12 (0.54) CA12CA1MMP2MMP9MMP8
Water SCHEMBL4754936 0.72 CA12 (0.53) CA12CA1MMP2MMP9MMP8
Water SCHEMBL4754935 0.72 CA12 (0.53) CA12CA1MMP2MMP9MMP8
Hydrochloric Acid SCHEMBL4754929 0.72 CA12 (0.53) CA12CA1MMP2MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed