Lithium Ion

Lithium Ion

SCHEMBL6433635

CC(C)[Si](Oc1ccc2cccc(C(=O)NCC(=O)[O-])c2c1)(C(C)C)C(C)C.[Li+]

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Lithium Ion. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 14/20 0.46
NQO2 P16083 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MTNR1B P49286 8/20 0.36
HTR2C P28335 2/20 0.35
HTR2B P41595 1/20 0.35
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6433632 0.88 MTNR1A (0.47) MTNR1ANQO2MEN1KMT2A
SCHEMBL6432839 0.88 MTNR1A (0.50) MTNR1ANQO2MEN1KMT2AMTNR1B
Lithium SCHEMBL6433640 0.88 MTNR1A (0.47) MTNR1ANQO2MEN1KMT2A
SCHEMBL6432988 0.79 NQO2 (0.47) MTNR1ANQO2MTNR1B
SCHEMBL6410573 0.79 MTNR1A (0.47) MTNR1ANQO2
SCHEMBL6582651 0.71 MTNR1A (0.52) MTNR1ANQO2MTNR1BHTR2CHTR2B
SCHEMBL6583218 0.68 HTR2A (0.49) MTNR1ANQO2MTNR1BHTR2CHTR2B
SCHEMBL6417161 0.68 HTR2A (0.35) MTNR1ANQO2MTNR1BHTR2CHTR2B
SCHEMBL7714927 0.67 TRPV1 (0.43) NQO2MEN1KMT2ATRPV1
SCHEMBL31670075 0.65 CYP2A6 (0.52) HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090011-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2005-04-06 EP disclosed
US-6410534-B1 ANTICANCER AGENTS MERCK & CO., INC. 2002-06-25 US disclosed
EP-1090011-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-11 EP disclosed
WO-2000001701-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed