SCHEMBL6433823

SCHEMBL6433823

NNC(=O)c1ccccc1NC(=O)Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.75
ALDH1A1 P00352 1/20 0.67
RXFP1 Q9HBX9 16/20 0.66
KDR P35968 1/20 0.65
MEN1 O00255 1/20 0.64
MAPT P10636 1/20 0.64
HTT P42858 1/20 0.64
RAB9A P51151 1/20 0.64
KMT2A Q03164 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1464137 0.89 GRIK1 (0.77) GRIK1RXFP1KDRMEN1MAPT
SCHEMBL9268782 0.86 RXFP1 (0.78) ALDH1A1RXFP1MAPTRAB9A
SCHEMBL1463217 0.86 GRIK1 (1.00) GRIK1RXFP1KDRMEN1MAPT
SCHEMBL17664319 0.85 KMT2A (0.82) GRIK1ALDH1A1RXFP1KDRMEN1
SCHEMBL6430550 0.83 GRIK1 (0.69) GRIK1RXFP1KDRMEN1MAPT
SCHEMBL23831539 0.83 MEN1 (0.64) GRIK1ALDH1A1MEN1MAPTHTT
SCHEMBL16127721 0.82 GRIK1 (0.75) GRIK1RXFP1KDRMEN1MAPT
SCHEMBL966454 0.81 ALDH1A1 (1.00) GRIK1ALDH1A1KDRMEN1MAPT
SCHEMBL5597699 0.81 KMT2A (0.90) GRIK1ALDH1A1KDRMEN1MAPT
SCHEMBL30101230 0.81 KMT2A (0.90) GRIK1ALDH1A1KDRMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050080112-A1 Compounds for use in disorders associated with mast cell or basophil acitvity POSEIDON PHARMACEUTICALS A/S (DK) 2005-04-14 US claimed
US-20050080112-A1 Compounds for use in disorders associated with mast cell or basophil acitvity POSEIDON PHARMACEUTICALS A/S (DK) 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080112-A1 Compounds for use in disorders associated with mast cell or basophil acitvity CPA3, HNMT, CMA1 GRIK1 655/4885ALDH1A1 327/4885RXFP1 2125/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.