SCHEMBL6434776

SCHEMBL6434776

COc1cc2c(Nc3cc(O)c(Br)cc3F)ccnc2cc1OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 6/20 0.59
FGFR1 P11362 4/20 0.59
EGFR P00533 6/20 0.51
KDR P35968 8/20 0.50
GAK O14976 2/20 0.48
RET P07949 4/20 0.47
KIF5B P33176 4/20 0.47
RAF1 P04049 1/20 0.46
BRAF P15056 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
SRC P12931 3/20 0.44
MET P08581 1/20 0.44
FGFR2 P21802 1/20 0.44
FGFR4 P22455 1/20 0.44
FGFR3 P22607 1/20 0.44
FLT4 P35916 1/20 0.44
BMPR1B O00238 1/20 0.43
EPHB6 O15197 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8509837 1.00 FLT1 (0.59) FLT1FGFR1EGFRKDRGAK
Hydrochloric Acid SCHEMBL6432639 0.99 FLT1 (0.58) FLT1FGFR1EGFRKDRGAK
SCHEMBL6433759 0.89 FLT1 (0.65) FLT1FGFR1EGFRKDRGAK
SCHEMBL6430998 0.89 FLT1 (0.75) FLT1FGFR1EGFRKDRRET
Hydrochloric Acid SCHEMBL6431427 0.88 FLT1 (0.74) FLT1FGFR1EGFRKDRRET
SCHEMBL27530363 0.85 EGFR (0.47) FLT1FGFR1EGFRKDRMET
Hydrochloric Acid SCHEMBL27532303 0.84 EGFR (0.46) FLT1FGFR1EGFRKDRMET
SCHEMBL6436593 0.83 MEN1 (0.43) FLT1FGFR1EGFRKDRRAF1
SCHEMBL6998899 0.82 FLT1 (0.74) FLT1FGFR1EGFRKDRSRC
SCHEMBL6433880 0.81 FLT1 (0.75) FLT1FGFR1EGFRKDRRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1252054-C Qinoline derivatives inhibiting effect of growth factors such as VEGF ZENECA LTD (GB) 2006-04-19 CN claimed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP claimed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US claimed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed