SCHEMBL6436802

SCHEMBL6436802

CC(C)(C)OC(=O)N(N)c1nc2nonc2nc1Nc1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.44
TP53 P04637 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
POLB P06746 1/20 0.44
CCR2 P41597 1/20 0.42
CCR5 P51681 1/20 0.42
CDK1 P06493 1/20 0.41
EGFR P00533 2/20 0.40
SRC P12931 1/20 0.40
GAA P10253 1/20 0.38
RECQL P46063 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
KDM1A O60341 1/20 0.38
MKNK1 Q9BUB5 1/20 0.37
PIM1 P11309 3/20 0.36
JAK2 O60674 2/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
HCK P08631 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6439454 0.88 GAA (0.45) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL6435667 0.87 MAPT (0.42) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL6431994 0.82 GAA (0.46) MAPTTP53SMN1; SMN2POLBGAA
SCHEMBL6416313 0.79 MAPT (0.47) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL6432336 0.77 SMN1; SMN2 (0.37) MAPTTP53SMN1; SMN2POLBGAA
SCHEMBL26035097 0.76 MAPK1 (0.46) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL26035099 0.74 STK17B (0.48) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL3056423 0.74 TP53 (0.63) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL26035439 0.73 TP53 (0.56) MAPTTP53SMN1; SMN2POLBCCR2
SCHEMBL6435103 0.71 HTT (0.33) POLBALDH1A1KDM4EKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005044270-A1 OXADIAZOLOPYRAZINE DERIVATIVES AS PHARMACEUTICALLY ACTIVE COMPOUNDS 4SC AG (DE) 2005-05-19 WO disclosed