SCHEMBL6437512

SCHEMBL6437512

O=C(Nc1ccccc1)c1ccc(OCc2ccc(Br)cc2)c(CCCCc2ncc[nH]2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 6/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
CASP3 P42574 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
POLB P06746 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
RXFP1 Q9HBX9 2/20 0.43
PARP1 P09874 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SCD O00767 1/20 0.42
SMPD1 P17405 1/20 0.42
MAPT P10636 2/20 0.42
FPR2 P25090 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4642686 0.93 NPC1 (0.45) LRRK2NPC1RAB9ACASP3SENP7
SCHEMBL4642232 0.87 RXRA (0.44) SMPD1
SCHEMBL5597306 0.80 SMPD1 (0.41) SMPD1HDAC1HDAC2
SCHEMBL5597311 0.80 RXRA (0.44) SMPD1FPR2
SCHEMBL6437508 0.75 FPR2 (0.47) LRRK2NPC1RAB9ACASP3SENP7
SCHEMBL4642071 0.75 LRRK2 (0.39) LRRK2NPC1RAB9APOLBKDM4E
SCHEMBL4642685 0.73 FPR2 (0.47) LRRK2NPC1RAB9ACASP3SENP7
SCHEMBL4640767 0.73 SMPD1 (0.41) SMPD1
SCHEMBL5597314 0.69 LRRK2 (0.37) LRRK2NPC1RAB9APOLBKDM4E
SCHEMBL11702689 0.69 CCR5 (0.48) NPC1RAB9ATAAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492515-A1 PHARMACEUTICAL COMPOSITION COMPRISING AN AROMATASE INHIBITOR AND AN ESTROGEN SUITABLE FOR HORMONE REPLACEMENT THERAPY FOR A MALE JENCAP RESEARCH LTD. (CA) 2005-01-05 EP disclosed
WO-2003082254-A1 PHARMACEUTICAL COMPOSITION COMPRISING AN AROMATASE INHIBITOR AND AN ESTROGEN SUITABLE FOR HORMONE REPLACEMENT THERAPY FOR A MALE JENCAP RESEARCH LTD. (CA) 2003-10-09 WO disclosed