SCHEMBL6438780

SCHEMBL6438780

CS(=O)(=O)c1ccc(-c2ccccc2-n2ccc(C(=O)O)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.50
PTGS1 P23219 2/20 0.44
JAK2 O60674 2/20 0.43
JAK3 P52333 1/20 0.43
AKR1C3 P42330 1/20 0.41
AKR1C1 Q04828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383807 0.85 ALDH1A1 (0.45) AKR1C3AKR1C1
SCHEMBL15754580 0.72 ALDH1A1 (0.54) AKR1C3AKR1C1
SCHEMBL3248259 0.72 PTGS2 (0.61) PTGS2PTGS1JAK2
SCHEMBL6789830 0.70 PTGS2 (0.68) PTGS2PTGS1
SCHEMBL2510446 0.70 IDO1 (0.42) PTGS2PTGS1AKR1C3AKR1C1
SCHEMBL3873486 0.69 CA12 (0.52) PTGS2PTGS1
SCHEMBL5502727 0.69 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL4638273 0.69 NOTUM (0.58) PTGS2
SCHEMBL1367745 0.69 MARS1 (0.44)
SCHEMBL22204516 0.68 GRM5 (0.40) AKR1C3AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed