SCHEMBL6439079

SCHEMBL6439079

CCCCCNCc1csc(C(C)C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
SLC6A3 Q01959 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP2D6 P10635 3/20 0.36
CYP2C19 P33261 3/20 0.36
ADORA2A P29274 1/20 0.36
LMNA P02545 1/20 0.36
ALDH1A1 P00352 4/20 0.35
TSHR P16473 1/20 0.35
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
STAT1 P42224 1/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15000428 0.79 KCNH2 (0.43) SLC6A3ADORA2AALDH1A1DRD2HTR2A
SCHEMBL28958748 0.75 HRH4 (0.38) HRH4HRH3SMN1; SMN2CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6090064 0.74 SLC6A3 (0.43) SLC6A3SMN1; SMN2ADORA2AALDH1A1DRD2
SCHEMBL28906001 0.73 SLC6A3 (0.43) SLC6A3SMN1; SMN2ADORA2AALDH1A1DRD2
SCHEMBL28958745 0.71 HPGD (0.56) HRH4HRH3LMNAALDH1A1TSHR
SCHEMBL28958749 0.70 HDAC1 (0.47) HRH4HRH3CYP1A2CYP2D6CYP2C19
Bicarbonate SCHEMBL29143008 0.69 ADORA2A (0.47) SLC6A3SMN1; SMN2ADORA2AALDH1A1DRD2
SCHEMBL18938015 0.68 SLC6A3 (0.41) SLC6A3CYP2D6CYP2C19ADORA2AALDH1A1
SCHEMBL16603147 0.68 SLC6A3 (0.46) SLC6A3ADORA2AALDH1A1DRD2HTR2A
SCHEMBL517979 0.67 KCNH2 (0.58) HRH4HRH3SMN1; SMN2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1509537-A2 CELLULAR ACCUMULATION OF PHOSPHONATE ANALOGS OF HIV PROTEASE INHIBITOR COMPOUNDS AND THE COMPOUNDS AS SUCH GILEAD SCIENCES, INC. (US) 2005-03-02 EP disclosed
WO-2003090690-A2 CELLULAR ACCUMULATION OF PHOSPHONATE ANALOGS OF HIV PROTEASE INHIBITOR COMPOUNDS AND THE COMPOUNDS AS SUCH GILEAD SCIENCES, INC. (US) 2003-11-06 WO disclosed