SCHEMBL6439335

SCHEMBL6439335

CC(C)(C)C1C[C]c2ccccc2N(Cc2nc(C(=O)N3CCC(CNc4ccccn4)CC3)cs2)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 9/20 0.41
NPY5R Q15761 1/20 0.37
EPHX1 P07099 1/20 0.34
EPHX2 P34913 1/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
NAMPT P43490 1/20 0.33
ITGB3 P05106 3/20 0.32
ITGAV P06756 3/20 0.32
ITGB1 P05556 2/20 0.32
ITGA2B P08514 2/20 0.32
ITGA5 P08648 2/20 0.32
ITGB5 P18084 2/20 0.32
NOS2 P35228 1/20 0.32
RBP4 P02753 1/20 0.32
PRMT5 O14744 1/20 0.32
PDE5A O76074 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE7A Q13946 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5028394 0.76 GRIN2B (0.40) GRIN2BNPY5REPHX1EPHX2CYP3A4
SCHEMBL5024033 0.75 GRIN2B (0.42) GRIN2BNPY5REPHX1EPHX2CYP3A4
SCHEMBL5879510 0.74 GRIN2B (0.41) GRIN2BNPY5REPHX1EPHX2CYP3A4
SCHEMBL3035919 0.66 GRIN2B (0.68) GRIN2BCYP3A4CYP2D6CYP2C9NOS2
SCHEMBL5028389 0.62 ITGB3 (0.41) ITGB3ITGAVITGA2BITGB5
SCHEMBL13118523 0.60 GRIN2B (0.57) GRIN2BITGB3ITGAVITGB1ITGA2B
SCHEMBL6442550 0.60 ALDH1A1 (0.32)
SCHEMBL5352852 0.60 GRIN2B (1.00) GRIN2BCYP3A4CYP2D6CYP2C9
SCHEMBL38662696 0.59 L3MBTL1 (0.49) NPY5REPHX1EPHX2NAMPTRBP4
Acetic Acid SCHEMBL5879702 0.58 ITGB3 (0.61) GRIN2BITGB3ITGAVITGB1ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286673-B8 LIGANDS OF INTEGRIN RECEPTORS ABBOTT GMBH & CO KG (DE) 2005-07-20 EP disclosed
EP-1286673-A2 LIGANDS OF INTEGRIN RECEPTORS Basf Aktiengesellschaft (DE) 2003-03-05 EP disclosed
WO-2001093840-A2 LIGANDS OF INTEGRIN RECEPTORS BASF AG (DE) 2001-12-13 WO disclosed