SCHEMBL6441183

SCHEMBL6441183

COC(=O)c1n[nH]c(-c2ccc(S(C)(=O)=O)cc2)c1C1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.43
KMT2A Q03164 1/20 0.41
ATR Q13535 1/20 0.40
PTGS1 P23219 1/20 0.39
GHSR Q92847 2/20 0.38
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
RAB9A P51151 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5150592 0.84 ALDH1A1 (0.36) KDM4ENPC1ALDH1A1RAB9A
SCHEMBL6444360 0.84 ALDH1A1 (0.36) KDM4ENPC1ALDH1A1RAB9A
SCHEMBL4957792 0.82 CCNB2 (0.41) PTGS2KMT2AATRPTGS1GHSR
SCHEMBL6438872 0.81 PTGS2 (0.47) PTGS2KMT2APTGS1GHSRBRD4
SCHEMBL6442228 0.77 PTGS2 (0.44) PTGS2PTGS1GHSRBRD4
SCHEMBL6439748 0.76 PTGS2 (0.44) PTGS2KMT2APTGS1GHSRBRD4
SCHEMBL6441485 0.75 PTGS2 (0.41) PTGS2PTGS1GHSR
SCHEMBL6438018 0.75 PTGS2 (0.43) PTGS2PTGS1GHSR
SCHEMBL6439880 0.75 PTGS2 (0.49) PTGS2PTGS1GHSR
SCHEMBL6439597 0.75 PTGS2 (0.41) PTGS2PTGS1GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed