SCHEMBL6444360

SCHEMBL6444360

COC(=O)c1n[nH]c(-c2ccc(SC)cc2)c1C1CCCCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.36
HPGD P15428 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.35
KDM4E B2RXH2 4/20 0.35
STAT3 P40763 1/20 0.35
HIF1A Q16665 1/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
RAB9A P51151 1/20 0.35
MAPT P10636 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
USP2 O75604 1/20 0.35
XBP1 P17861 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5150592 1.00 ALDH1A1 (0.36) ALDH1A1HPGDSMN1; SMN2LMNAGAA
SCHEMBL6441183 0.84 PTGS2 (0.43) ALDH1A1KDM4ERAB9ANPC1
SCHEMBL4960913 0.82 GSK3B (0.41) ALDH1A1HPGDSMN1; SMN2LMNAKDM4E
SCHEMBL6440473 0.78 GAA (0.43) ALDH1A1HPGDSMN1; SMN2LMNAGAA
SCHEMBL6441497 0.74 ALDH1A1 (0.53) ALDH1A1HPGDSMN1; SMN2LMNAGAA
SCHEMBL6442323 0.74 GAA (0.40) ALDH1A1HPGDSMN1; SMN2LMNAGAA
SCHEMBL6441245 0.73 MAPT (0.45) ALDH1A1HPGDSMN1; SMN2LMNAKDM4E
SCHEMBL6441172 0.73 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2LMNAGAAKDM4E
SCHEMBL6440359 0.73 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2LMNAKDM4ESTAT3
SCHEMBL6439608 0.73 MAPT (0.45) ALDH1A1HPGDSMN1; SMN2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed