SCHEMBL6441263

SCHEMBL6441263

Brc1ccc2c(c1)C(c1ccc(Oc3ccccc3)cc1)(c1ccc(Oc3ccccc3)cc1)c1cc(Br)ccc1-2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.42
MAOA P21397 5/20 0.41
MAOB P27338 4/20 0.41
LTA4H P09960 3/20 0.39
TSHR P16473 1/20 0.39
GSTP1 P09211 1/20 0.39
MCL1 Q07820 2/20 0.38
PGR P06401 1/20 0.38
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
NR1H2 P55055 1/20 0.36
BAX Q07812 1/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14823249 1.00 PDK2 (0.42) PDK2MAOAMAOBLTA4HTSHR
SCHEMBL13129740 0.95 PDK2 (0.43) PDK2MAOAMAOBLTA4HTSHR
SCHEMBL13129739 0.92 PDK2 (0.37) PDK2MAOAMAOBLTA4HTSHR
SCHEMBL21793205 0.89 LTA4H (0.46) PDK2MAOAMAOBLTA4HTSHR
SCHEMBL22197320 0.86 LTA4H (0.50) PDK2MAOAMAOBLTA4HTSHR
SCHEMBL22197292 0.86 ALDH1A1 (0.40) PDK2MAOAMAOBMCL1PGR
SCHEMBL21793629 0.86 PDK2 (0.41) PDK2MAOAMAOBPGRMAPT
SCHEMBL1307887 0.84 PDK2 (0.47) PDK2MAPTKDM4EMEN1LMNA
SCHEMBL29540116 0.84 PDK2 (0.47) PDK2MAPTKDM4EMEN1LMNA
SCHEMBL23713945 0.83 PDK2 (0.39) PDK2MAOAMAOBPGRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8410243-B2 Aromatic ether-containing fluorene monomers, processes for their preparation and polymerization thereof THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2013-04-02 US disclosed
US-20100240856-A1 Aromatic Ether-Containing Fluorene Monomers, Processes for their Preparation and Polymerization Thereof THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2010-09-23 US disclosed
US-6900285-B2 Fluorene-containing polymers and compounds useful in the preparation thereof DOW GLOBAL TECHNOLOGIES INC. (US) 2005-05-31 US disclosed
US-20030208032-A1 Fluorene-containing polymers and compounds useful in the preparation thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-11-06 US disclosed
US-6514632-B1 Electroluminescent films and coatings for light emitting diodes; efficiency DOW GLOBAL TECHNOLOGIES INC. 2003-02-04 US disclosed
US-6512083-B1 Film prepared from the polymers of this invention. this invention is a light-emitting diode comprised of one or more layers of polymer films, at least one of which is derived from the oligomers and polymers of the invention. DOW GLOBAL TECHNOLOGIES INC. 2003-01-28 US disclosed
US-6362310-B1 LIGHT EMITTING POLYMER SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-03-26 US disclosed
US-6255449-B1 PROCESS FOR PREPARING POLYMERS HAVING AT LEAST THREE FLUORENE GROUPS IN BACKBONE, WHICH COMPRISES HEATING 2,7-DIHALO-9-SUBSTITUTED FLUORENES UNDER REACTION CONDITIONS SUFFICIENT TO FORM SAID POLYMERS THE DOW CHEMICAL COMPANY 2001-07-03 US disclosed
US-6169163-B1 NOVEL 2,7-DIHALOFLUORENES SUBSTITUTED AT 9-POSITION THE DOW CHEMICAL COMPANY 2001-01-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240856-A1 Aromatic Ether-Containing Fluorene Monomers, Processes for their Preparation and Polymerization Thereof TYR, PAH, AFF4 PDK2 2716/4885MAOA 638/4885MAOB 501/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.