SCHEMBL6442811

SCHEMBL6442811

O=C(CN1C(=O)CC[C]c2ccccc21)NCC1CCC(NC(=O)NCc2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.45
EPHX1 P07099 1/20 0.44
HPGD P15428 1/20 0.44
DRD4 P21917 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ITGB3 P05106 3/20 0.42
ITGAV P06756 3/20 0.42
NPY5R Q15761 6/20 0.41
TSHR P16473 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5025462 0.81 ITGB3 (0.63) MAPK1EPHX1HPGDDRD4NPSR1
SCHEMBL20911011 0.70 EPHX1 (0.84) EPHX1HPGDDRD4TSHRNPC1
SCHEMBL6439601 0.70 ITGB3 (0.54) MAPK1ITGB3ITGAVTSHRNPC1
SCHEMBL23349229 0.69 EPHX1 (0.73) EPHX1HPGDDRD4TSHRNPC1
SCHEMBL6445537 0.69 ITGB3 (0.49) MAPK1ITGB3ITGAVTSHRL3MBTL1
SCHEMBL6444182 0.68 ITGB3 (0.56) MAPK1HPGDITGB3ITGAVNPC1
SCHEMBL5028143 0.67 EPHX1 (0.69) EPHX1HPGDDRD4TSHRNPC1
SCHEMBL5318930 0.67 EPHX1 (0.69) EPHX1HPGDDRD4TSHRNPC1
SCHEMBL5028140 0.67 EPHX1 (0.69) EPHX1HPGDDRD4TSHRNPC1
SCHEMBL6440168 0.67 ITGB3 (0.67) MAPK1ITGB3ITGAVL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286673-B8 LIGANDS OF INTEGRIN RECEPTORS ABBOTT GMBH & CO KG (DE) 2005-07-20 EP disclosed
EP-1286673-A2 LIGANDS OF INTEGRIN RECEPTORS Basf Aktiengesellschaft (DE) 2003-03-05 EP disclosed
WO-2001093840-A2 LIGANDS OF INTEGRIN RECEPTORS BASF AG (DE) 2001-12-13 WO disclosed