SCHEMBL6445446

SCHEMBL6445446

N#CCNC(=O)C(CNC(=O)c1cccc(C(F)(F)F)c1)c1csc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 8/20 0.55
GPR139 Q6DWJ6 1/20 0.46
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
NPC1 O15118 1/20 0.42
CTSS P25774 2/20 0.41
CTSK P43235 2/20 0.41
TACR1 P25103 1/20 0.41
LMNA P02545 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 1/20 0.40
TP53BP1 Q12888 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822574 0.91 CTSL (0.44) CTSLGPR139ALDH1A1POLBNPC1
SCHEMBL6448205 0.88 CTSL (0.47) CTSLCTSSCTSK
SCHEMBL6446814 0.85 CTSL (0.41) CTSLCTSSCTSK
SCHEMBL6446641 0.83 CTSL (0.64) CTSLGPR139ALDH1A1POLBNPC1
SCHEMBL6447552 0.80 CTSK (0.42) CTSLCTSSCTSK
SCHEMBL6020607 0.80 CTSL (0.64) CTSLCTSSCTSKTACR1
SCHEMBL6821937 0.79 CTSK (0.43) CTSLALDH1A1POLBNPC1CTSS
SCHEMBL6021296 0.79 CTSL (0.38) CTSLNPC1CTSSCTSKRAB9A
SCHEMBL6021888 0.79 CTSK (0.44) CTSLPOLBCTSSCTSK
SCHEMBL6446486 0.79 CTSK (0.41) CTSLALDH1A1NPC1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed